专利检索 ipc:"C07D209/196" 第 1 页

1.

发明授权
5-halo-tryptamine derivatives used as ligands on the 5-HT6 and/or 5-HT7 serotonin receptors 失效
标题翻译：用作5-HT6和/或5-HT7血清素受体的配体的5-卤素 - 色胺衍生物

公开(公告)号：US07098233B2

公开(公告)日：2006-08-29

申请号：US10481433

申请日：2002-06-17

申请人： Maria Assunta Di Cesare , Patrizia Minetti , Giorgio Tarzia , Gilberto Spadoni

发明人： Maria Assunta Di Cesare , Patrizia Minetti , Giorgio Tarzia , Gilberto Spadoni

IPC分类号： A61K31/405 , C07D209/196

CPC分类号： C07D209/16 , A61K31/405

摘要： Compounds of Formula (I): (I); wherein: R1 and R2 either the same or different, are H or linear or branched C1–C6 alkyl; R3=linear or branched C1–C6 alkyl; R4=halogen, and pharmaceutically acceptable salts thereof are useful as active ingredients in the preparation of medicaments used as ligands of the 5-HT6 and/or 5-HT7 serotoninergic receptors.

摘要翻译： 式（I）的化合物：（I）; 其中：R 1和R 2相同或不同，为H或直链或支链C 1 -C 6 - 烷基; R 3 =直链或支链C 1 -C 6烷基; R 4 =卤素及其药学上可接受的盐可用作制备用作5-HT 6和/或5-HT 6配体的药物的活性成分， 5-羟色胺能受体。