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1.IMPROVED PROCESS FOR PREPARATION OF SAXAGLIPTIN AND ITS SALTS 审中-公开
Title translation: 改进萨伐他汀及其盐的制备方法公开(公告)号:WO2013175395A3
公开(公告)日:2014-01-30
申请号:PCT/IB2013054167
申请日:2013-05-21
Applicant: REDDYS LAB LTD DR
Inventor: VARANASI GANESH , MACHARLA PRABHAKAR , VEMPATI CHANDRASEKHAR , BANDICHHOR RAKESHWAR , DAHANUKAR VILAS HARESHWAR , IQBAL JAVED , ORUGANTI SRINIVAS , RAPOLU RAJESH KUMAR , NARIYAM MUNASWAMY SEKHAR , NETI SRINIVASAN
IPC: C07D209/02 , A61K31/403 , C07C13/615 , C07D209/52
CPC classification number: C07D209/52
Abstract: Improved processes for preparing saxagliptin or its salt and intermediates thereof are provided.
Abstract translation: 提供了制备沙格列汀或其盐及其中间体的改进方法。
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公开(公告)号:WO2010014883A3
公开(公告)日:2010-05-14
申请号:PCT/US2009052376
申请日:2009-07-31
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR , CHERUKUPALLY PRAVEEN , VUJJINI SATISH KUMAR , VARANASI GANESH , KANDALA SREENADHA CHARYULU , AREVELI SRINIVAS , TIRUMALARAJU SATYANARAYANA RAJ
Inventor: CHERUKUPALLY PRAVEEN , VUJJINI SATISH KUMAR , VARANASI GANESH , KANDALA SREENADHA CHARYULU , AREVELI SRINIVAS , TIRUMALARAJU SATYANARAYANA RAJU
IPC: C07D405/04 , A61K31/53 , C07D251/42 , C07D405/02
CPC classification number: C07H17/02 , A61K31/53 , C07D405/04 , C07H13/12 , C07H19/12
Abstract: Processes for preparing azacitidine. Further included are processes for the preparation of crystalline azacitidine crystalline Form (I) and mixtures of azacitidine crystalline Forms (I) and (II).
Abstract translation: 制备阿扎胞苷的方法。 还包括制备结晶阿扎胞苷结晶形式(I)和阿扎胞苷结晶形式(I)和(II)的混合物的方法。
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