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公开(公告)号：WO2015101957A3
公开(公告)日：2015-11-19
申请号：PCT/IB2015050075
申请日：2015-01-05
发明人： BHAVAR PRASHANT KASHINATH , VAKKALANKA SWAROOP KUMAR VENKATA SATYA , VISWANADHA SRIKANT , SWAROOP MERIKAPUDI GAYATRI , BABU GOVINDARAJULU
IPC分类号： C07D417/06 , A61K31/433 , A61P35/00 , A61P37/00 , C07D285/135 , C07D417/08 , C07D417/14
CPC分类号： C07D417/14 , A61K31/433 , A61K31/44 , A61K31/4439 , A61K31/444 , A61K31/4545 , A61K31/4965 , A61K31/497 , A61K31/501 , A61K31/505 , A61K31/506 , A61K45/06 , C07D213/75 , C07D239/42 , C07D241/20 , C07D285/135 , C07D401/04 , C07D401/12 , C07D417/06 , C07D417/08
摘要： The present disclosure provides compounds of formula (I) to (III) as glutaminase inhibitors, methods of preparing them, pharmaceutical compositions containing them and methods of treatment, prevention and/or amelioration of diseases or disorders involving glutamine.
摘要翻译： 本公开内容提供式（I）至（III）的化合物作为谷氨酰胺酶抑制剂，其制备方法，含有它们的药物组合物以及治疗，预防和/或改善涉及谷氨酰胺的疾病或病症的方法。
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2.发明申请NOVEL 3,5-DISUBSTITUED-3H-IMIDAZO[4,5-B]PYRIDINE AND 3,5- DISUBSTITUED -3H-[1,2,3]TRIAZOLO[4,5-B] PYRIDINE COMPOUNDS AS MODULATORS OF C-MET PROTEIN KINASES 审中-公开作为C-MET调节剂的新的3,5-二取代的-3H-咪唑并[4,5-B]吡啶和3,5-二取代的-3H- [1,2,3]三唑并[4,5-B]吡啶化合物 蛋白激酶
公开(公告)号：WO2013144737A3
公开(公告)日：2013-12-05
申请号：PCT/IB2013051577
申请日：2013-02-27
发明人： VAKKALANKA SWAROOP KUMAR VENKATA SATYA , NAGARATHNAM DHANAPALAN , VISWANADHA SRIKANT , MUTHUPPALANIAPPAN MEYYAPPAN , BABU GOVINDARAJULU , BHAVAR PRASHANT K
IPC分类号： C07D471/04 , A61K31/437 , A61K31/4709 , A61P35/00
CPC分类号： C07D471/04 , A61K31/437 , A61K31/4709 , A61K45/06
摘要： The present invention provides compounds useful as C-met protein kinase modulators, methods of preparing them, pharmaceutical compositions containing them and methods of treatment, prevention and/or amelioration of C-met kinase mediated diseases or disorders with them.
摘要翻译： 本发明提供可用作C-met蛋白激酶调节剂的化合物，其制备方法，含有它们的药物组合物以及用它们治疗，预防和/或缓解C-met激酶介导的疾病或病症的方法。
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3.发明申请NOVEL 3,5-DISUBSTITUED-3H-IMIDAZO[4,5-B]PYRIDINE AND 3,5- DISUBSTITUED -3H-[1,2,3]TRIAZOLO[4,5-B] PYRIDINE COMPOUNDS AS MODULATORS OF PROTEIN KINASES 审中-公开新的3,5-取代-3H-咪唑并[4,5-B]吡啶和3,5-分解的-3H- [1,2,3]三唑并[4,5-B]吡啶化合物作为蛋白激酶的调节剂
公开(公告)号：WO2011145035A8
公开(公告)日：2012-06-21
申请号：PCT/IB2011052120
申请日：2011-05-13
申请人： INCOZEN THERAPEUTICS PVT LTD , RHIZEN PHARMACEUTICALS SA , MUTHUPPALANIAPPAN MEYYAPPAN , VISWANADHA SRIKANT , BABU GOVINDARAJULU , VAKKALANKA SWAROOP K V S
发明人： MUTHUPPALANIAPPAN MEYYAPPAN , VISWANADHA SRIKANT , BABU GOVINDARAJULU , VAKKALANKA SWAROOP K V S
IPC分类号： C07D471/04 , A61K31/437 , A61K31/4709 , A61P35/00
CPC分类号： C07D471/04 , A61K31/437 , A61K31/4709 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K45/06 , G01N33/5011 , G01N2500/10
摘要： The present invention provides, inter alia, compounds of formula ??,??? and III as protein kinase modulators, methods of preparing them, pharmaceutical compositions containing them and methods of treatment, prevention and/or amelioration of kinase mediated diseases or disorders with them.
摘要翻译： 本发明尤其提供式Ⅻ， 和III作为蛋白激酶调节剂，其制备方法，含有它们的药物组合物以及用它们治疗，预防和/或改善激酶介导的疾病或病症的方法。
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公开(公告)号：WO2015101958A2
公开(公告)日：2015-07-09
申请号：PCT/IB2015050076
申请日：2015-01-05
发明人： BHAVAR PRASHANT KASHINATH , VAKKALANKA SWAROOP KUMAR VENKATA SATYA , VISWANADHA SRIKANT , SWAROOP MERIKAPUDI GAYATRI , BABU GOVINDARAJULU
IPC分类号： C07D417/06 , A61K31/433 , A61P35/00 , A61P37/00 , C07D285/135 , C07D417/08 , C07D417/14
CPC分类号： C07D417/14 , A61K31/433 , A61K31/44 , A61K31/4439 , A61K31/444 , A61K31/4545 , A61K31/4965 , A61K31/497 , A61K31/501 , A61K31/505 , A61K31/506 , A61K45/06 , C07D213/75 , C07D239/42 , C07D241/20 , C07D285/135 , C07D401/04 , C07D401/12 , C07D417/06 , C07D417/08
摘要： The present disclosure provides compounds of formula (I) to (III) as glutaminase inhibitors, methods of preparing them, pharmaceutical compositions containing them and methods of treatment, prevention and/or amelioration of diseases or disorders involving glutamine.
摘要翻译： 本公开内容提供式（I）至（III）的化合物作为谷氨酰胺酶抑制剂，其制备方法，含有它们的药物组合物以及治疗，预防和/或改善涉及谷氨酰胺的疾病或病症的方法。
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公开(公告)号：WO2011055215A3
公开(公告)日：2011-08-25
申请号：PCT/IB2010002804
申请日：2010-11-03
申请人： INCOZEN THERAPEUTICS PVT LTD , RHIZEN PHARMACEUTICALS SA , MUTHUPPALANIAPPAN MEYYAPPAN , VISWANADHA SRIKANT , BABU GOVINDARAJULU , VAKKALANKA SWAROOP KUMAR V S
发明人： MUTHUPPALANIAPPAN MEYYAPPAN , VISWANADHA SRIKANT , BABU GOVINDARAJULU , VAKKALANKA SWAROOP KUMAR V S
IPC分类号： C07D311/34 , A61K31/519 , A61K31/52 , A61P35/00 , A61P37/06 , C07D405/06 , C07D487/04
CPC分类号： C07D311/36 , A61K31/352 , A61K31/4178 , A61K31/4184 , A61K31/437 , A61K31/519 , A61K31/52 , A61K31/522 , A61K31/5377 , A61K45/06 , C07D405/06 , C07D413/10 , C07D413/14 , C07D471/04 , C07D473/08 , C07D473/34 , C07D473/38 , C07D473/40 , C07D487/04
摘要： The present invention provides PL3K protein kinase modulators, methods of preparing them, pharmaceutical compositions containing them and methods of treatment, prevention and/or amelioration of kinase mediated diseases or disorders with them.
摘要翻译： 本发明提供了PL3K蛋白激酶调节剂，其制备方法，含有它们的药物组合物以及用它们治疗，预防和/或改善激酶介导的疾病或病症的方法。
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