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发明公开
CN101304987A 作为人类免疫缺陷病毒蛋白酶抑制剂的氨基苯基磺酰胺衍生物 失效 - 权利终止 转让

作为人类免疫缺陷病毒蛋白酶抑制剂的氨基苯基磺酰胺衍生物
摘要：
本发明涉及经取代的氨基苯基磺酰胺化合物及衍生物，它们作为蛋白酶抑制剂的用途，特别是作为广效HIV蛋白酶抑制剂，这些化合物以及药学组合物的制备方法以及含有这些化合物的诊断试剂盒。本发明亦涉及该经取代氨基苯基磺酰胺化合物及衍生物与另一抗逆转录病毒剂的组合。其进一步有关于它们在分析中作为参考化合物或作为试剂的用途。
摘要（英）：

The present invention concerns substituted aminophenylsulfonamide compounds and derivatives, their use as protease inhibitors, in particular as broadspectrum HIV protease inhibitors, processes for their preparation as well as pharmaceutical compositions and diagnostic kits comprising them. The present invention also concerns combinations of the present substituted aminophenylsulfonamide compounds and derivatives with another anti-retroviral agent. It further relates to their use in assays as reference compounds or as reagents.

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