发明公开
EP0393538A2 Thiazetoquinoline-3-Carboxylic acid derivative, method for preparation thereof, and a pharmaceutical composition comprising the same
失效
Thiazetochinolin -3-羧酸衍生物，它们的制备方法和含有药物制备方法。
- 专利标题： Thiazetoquinoline-3-Carboxylic acid derivative, method for preparation thereof, and a pharmaceutical composition comprising the same
- 专利标题（中）： Thiazetochinolin -3-羧酸衍生物，它们的制备方法和含有药物制备方法。
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申请号： EP90107124.1申请日： 1990-04-13
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公开(公告)号： EP0393538A2公开(公告)日： 1990-10-24
- 发明人: Itoh, Yasuo , Kato, Hideo , Koshinaka, Eiichi , Ogawa, Nobuo , Yagi, Noriyuki , Yoshida, Toshihiko , Suzuki, Tomio
- 申请人： HOKURIKU PHARMACEUTICAL CO., LTD.
- 申请人地址： 1-Chome, 3-14, Tatekawacho, Katsuyama-shi Fukui-ken 911 JP
- 专利权人： HOKURIKU PHARMACEUTICAL CO., LTD.
- 当前专利权人： HOKURIKU PHARMACEUTICAL CO., LTD.
- 当前专利权人地址： 1-Chome, 3-14, Tatekawacho, Katsuyama-shi Fukui-ken 911 JP
- 代理机构： Werner, Hans-Karsten, Dr.Dipl.-Chem.
- 优先权： JP96328/89 19890418; JP223217/89 19890831; JP264840/89 19891016
- 主分类号： C07D513/04
- IPC分类号： C07D513/04 ; A61K31/435
摘要：
A thiazetoquinoline-3-carboxylic acid derivative represented by the general formula (I)
wherein R₁ is a hydrogen atom or a lower alkyl group; R₂ is a fluorine atom or a chlorine atom; R₃ is a hydrogen atom, a lower alkyl group, a lower alkanoyl group, a halogenated lower alkanoyl, or alkoxycarbonyl group; and R₄ is a hydrogen atom or a lower alkyl group, and a pharmacologically acceptable salt thereof, a process for preparation thereof, a pharmaceutical composition comprising the same, and a method for the treatment of an infectious disease by administering the same, are disclosed.
wherein R₁ is a hydrogen atom or a lower alkyl group; R₂ is a fluorine atom or a chlorine atom; R₃ is a hydrogen atom, a lower alkyl group, a lower alkanoyl group, a halogenated lower alkanoyl, or alkoxycarbonyl group; and R₄ is a hydrogen atom or a lower alkyl group, and a pharmacologically acceptable salt thereof, a process for preparation thereof, a pharmaceutical composition comprising the same, and a method for the treatment of an infectious disease by administering the same, are disclosed.
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