发明公开
- 专利标题: 6-HETEROARYLPHENANTHRIDINES
- 专利标题(中): 6- HETEROARYLPHENANTHRIDINES
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申请号: EP01962844.5申请日: 2001-07-07
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公开(公告)号: EP1303506A1公开(公告)日: 2003-04-23
- 发明人: BUNDSCHUH, Daniela , FLOCKERZI, Dieter , GRUNDLER, Gerhard , HATZELMANN, Armin , KLEY, Hans-Peter , WEINBRENNER, Steffen , GUTTERER, Beate
- 申请人: Byk Gulden Lomberg Chemische Fabrik GmbH
- 申请人地址: Byk-Gulden-Str. 2 78467 Konstanz DE
- 专利权人: Byk Gulden Lomberg Chemische Fabrik GmbH
- 当前专利权人: Byk Gulden Lomberg Chemische Fabrik GmbH
- 当前专利权人地址: Byk-Gulden-Str. 2 78467 Konstanz DE
- 优先权: EP00115352 20000714
- 国际公布: WO02006270 20020124
- 主分类号: C07D401/04
- IPC分类号: C07D401/04 ; A61K31/473 ; A61P11/06 ; C07D405/04 ; C07D409/04 ; C07D413/04 ; C07D417/04
摘要:
Compounds of the formula I, in which Het is an unsubstituted or R6-and/or R7-sustituted pyrrolyl, furanyl, thiophenyl, pyrazolyl, imidazolyl, oxazolyl, isoxazolyl, thiazolyl, isothiazolyl, thiadiazolyl, pyrimidinyl, pyrazinyl or pyridazinyl radical, or an unsubstituted or R6-and/or R7-substituted fused bi-or tricyclic ring system comprising at least one aromatic ring and up to 4 heteroatoms-selected from the group consisting of O(oxygen), S(sulphur) or N(nitrogen)-which is bonded to the phenanthridinyl radical via one of the rings comprising one or more heteroatoms, areactive PDE4 inhibitors.
公开/授权文献
- EP1303506B1 6-HETEROARYLPHENANTHRIDINES 公开/授权日:2005-02-02
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