发明公开
EP1389618A1 PYRAZOLO 1,5-A]PYRIDINES AND MEDICINES CONTAINING THE SAME
有权
吡咯唑酮1,5-A PYRIDINE IN DIESE ENTHALTENDE ARZNEIMITTEL
- 专利标题: PYRAZOLO 1,5-A]PYRIDINES AND MEDICINES CONTAINING THE SAME
- 专利标题(中): 吡咯唑酮1,5-A PYRIDINE IN DIESE ENTHALTENDE ARZNEIMITTEL
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申请号: EP02720608.5申请日: 2002-04-25
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公开(公告)号: EP1389618A1公开(公告)日: 2004-02-18
- 发明人: HIBI, Shigeki , KIKUCHI, Koichi , HOSHINO, Yorihisa , SOEJIMA, Motohiro , YOSHIUCHI, Tatsuya , SHIN, Kogyoku , ONO, Mutsuko , TAKAHASHI, Yoshinori , SHIBATA, Hisashi , INO, Mitsuhiro , HIRAKAWA, Tetsuya
- 申请人: Eisai Co., Ltd.
- 申请人地址: 6-10, Koishikawa 4-chome, Bunkyo-ku Tokyo 112-8088 JP
- 专利权人: Eisai Co., Ltd.
- 当前专利权人: Eisai Co., Ltd.
- 当前专利权人地址: 6-10, Koishikawa 4-chome, Bunkyo-ku Tokyo 112-8088 JP
- 代理机构: HOFFMANN EITLE
- 优先权: JP2001133207 20010427
- 国际公布: WO2002088121 20021107
- 主分类号: C07D471/04
- IPC分类号: C07D471/04 ; A61K31/437 ; A61K31/444 ; A61P3/04 ; A61P3/10 ; A61P9/00 ; A61P9/10 ; A61P15/00 ; A61P19/00 ; A61P25/08 ; A61P25/18 ; A61P25/22 ; A61P25/24 ; A61P25/28 ; A61P37/08 ; A61P11/00 ; A61P43/00
摘要:
Compounds represented by the general formula:
[wherein R 1 represents methoxy, ethyl, methylthio, etc., R 2 , R 3 and R 4 each represent hydrogen, a halogen, etc., R 5 and R 6 each represent -X 5 -X 6 -X 7 (wherein X 5 represents a single bond or -CO-, X 6 represents a single bond, -NR 3a , etc. and X 7 and R 3a each represent hydrogen, C 1-10 alkyl, etc.), and Ar represents phenyl, pyridyl, etc.], salts thereof and hydrates of the foregoing.
[wherein R 1 represents methoxy, ethyl, methylthio, etc., R 2 , R 3 and R 4 each represent hydrogen, a halogen, etc., R 5 and R 6 each represent -X 5 -X 6 -X 7 (wherein X 5 represents a single bond or -CO-, X 6 represents a single bond, -NR 3a , etc. and X 7 and R 3a each represent hydrogen, C 1-10 alkyl, etc.), and Ar represents phenyl, pyridyl, etc.], salts thereof and hydrates of the foregoing.
公开/授权文献
- EP1389618B1 PYRAZOLO 1,5-A PYRIDINES AND MEDICINES CONTAINING THE SAME 公开/授权日:2011-06-15
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