发明公开
EP2054053A1 BIPHENYL SUBSTITUIERTE SPIROTETRONSÄUREN UND IHRE VERWENDUNG ZUR BEHANDLUNG RETROVIRALER ERKRANKUNGEN
审中-公开
联苯取代SPIROTETRONSÄUREN及其用于治疗病毒性疾病RETRO
- 专利标题: BIPHENYL SUBSTITUIERTE SPIROTETRONSÄUREN UND IHRE VERWENDUNG ZUR BEHANDLUNG RETROVIRALER ERKRANKUNGEN
- 专利标题(英): Biphenyl substituted spirotetronic acids and their use for the treatment of retroviral disorders
- 专利标题(中): 联苯取代SPIROTETRONSÄUREN及其用于治疗病毒性疾病RETRO
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申请号: EP07801624.3申请日: 2007-08-13
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公开(公告)号: EP2054053A1公开(公告)日: 2009-05-06
- 发明人: HEIMBACH, Dirk , TERSTEEGEN, Adrian , THEDE, Kai , WELKER, Reinhold , FAST, Beate , PAESSENS, Arnold , DITTMER, Frank , SCHOHE-LOOP, Rudolf , HARRENGA, Axel , HILLISCH, Alexander , HENNINGER, Kerstin , HÜBSCH, Walter , BAUSER, Marcus , PAULSEN, Daniela , BIRKMANN, Alexander , BRETSCHNEIDER, Thomas , FISCHER, Reiner , GRESCHAT, Susanne , URBAN, Andreas , WILDUM, Steffen
- 申请人: AiCuris GmbH & Co. KG
- 申请人地址: Friedrich-Ebert-Strasse 475 42117 Wuppertal DE
- 专利权人: AiCuris GmbH & Co. KG
- 当前专利权人: AiCuris GmbH & Co. KG
- 当前专利权人地址: Friedrich-Ebert-Strasse 475 42117 Wuppertal DE
- 代理机构: Scheuermann, Erik
- 优先权: DE102006039912 20060825
- 国际公布: WO2008022725 20080228
- 主分类号: A61K31/343
- IPC分类号: A61K31/343 ; C07D307/94 ; C07D405/12 ; C07D407/10 ; C07D491/10 ; C07D493/10 ; C07D495/10
摘要:
The present invention relates to novel substituted spirotetronic acids (I) in which R1 and R2, together with the carbon atom to which they are bonded, form a group of the formula (1), (2), (3) or (4), where * is the carbon atom to which R1 and R2 are bonded, to processes for their preparation, their use for the treatment and/or prophylaxis of diseases, and their use for producing medicaments for the treatment and/or prophylaxis of diseases, in particular of retroviral disorders, in people and/or animals.
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