发明公开
EP2356106A1 BIARYL SPIROAMINOOXAZOLINE ANALOGUES AS ALPHA2C ADRENERGIC RECEPTOR MODULATORS
审中-公开
作为ALPHA2C肾上腺素能受体调节剂的双酰基螺旋酰胺肟类似物
- 专利标题： BIARYL SPIROAMINOOXAZOLINE ANALOGUES AS ALPHA2C ADRENERGIC RECEPTOR MODULATORS
- 专利标题（中）： 作为ALPHA2C肾上腺素能受体调节剂的双酰基螺旋酰胺肟类似物
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申请号： EP09793312.1申请日： 2009-10-06
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公开(公告)号： EP2356106A1公开(公告)日： 2011-08-17
- 发明人: MCCORMICK, Kevin D. , DONG, Li , BOYCE, Christopher W , DE LERA RUIZ, Manuel , FEVRIER, Salem , WU, Jie , ZHENG, Junying , YU, Younong , CHAO, Jianhua , WON, Walter S. , RAO, Ashwin U. , KUANG, Rongze , TING, Pauline C. , HUANG, Xianhai , SHAO, Ning , PALANI, Anandan , BERLIN, Michael Y. , ASLANIAN, Robert G.
- 申请人： Schering Corporation
- 申请人地址： 2000 Galloping Hill Road Kenilworth, NJ 07033-0530 US
- 专利权人： Schering Corporation
- 当前专利权人： Schering Corporation
- 当前专利权人地址： 2000 Galloping Hill Road Kenilworth, NJ 07033-0530 US
- 代理机构： Buchan, Gavin MacNicol
- 优先权： US103409P 20081007
- 国际公布： WO2010042473 20100415
- 主分类号： C07D401/10
- IPC分类号： C07D401/10 ; C07D403/10 ; C07D405/10 ; C07D409/10 ; C07D413/10 ; C07D417/10 ; C07D235/02 ; C07D263/52 ; C07D498/10 ; C07D519/00 ; A61K31/4184 ; A61K31/4188 ; A61K31/424 ; A61P11/02
摘要：
In its many embodiments, the present invention provides a novel class of biaryi spiroaminooxazoline analogues as modulators of α2C adrenergic receptor agonists, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more conditions associated with the α2C adrenergic receptors using such compounds or pharmaceutical compositions.
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