发明公开
EP2484679A3 N3-heteroaryl substituted triazoles and n5-heteroaryl substitued triazoles useful as axl inhibitors
有权
N3-杂芳基取代的三唑和n5-杂芳基取代的三唑，可用作AX1抑制剂
- 专利标题： N3-heteroaryl substituted triazoles and n5-heteroaryl substitued triazoles useful as axl inhibitors
- 专利标题（中）： N3-杂芳基取代的三唑和n5-杂芳基取代的三唑，可用作AX1抑制剂
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申请号： EP12002451.8申请日： 2007-12-28
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公开(公告)号： EP2484679A3公开(公告)日： 2012-10-10
- 发明人: Goff, Ding , Zhang, Jing , Singh, Rajinder , Holland, Sacha , Yu, Jiaxin , Heckrodt, Thilo , Ding, Pingyu , Litvak, Joane
- 申请人： Rigel Pharmaceuticals, Inc.
- 申请人地址： 1180 Veterans Boulevard South San Francisco, CA 94080 US
- 专利权人： Rigel Pharmaceuticals, Inc.
- 当前专利权人： Rigel Pharmaceuticals, Inc.
- 当前专利权人地址： 1180 Veterans Boulevard South San Francisco, CA 94080 US
- 代理机构： Grünecker, Kinkeldey, Stockmair & Schwanhäusser
- 优先权： US882875P 20061229; US975443P 20070926
- 主分类号： C07D405/12
- IPC分类号： C07D405/12 ; C07D405/14 ; C07D413/14 ; C07D471/04 ; C07D495/04 ; C07D519/00 ; C07D487/04 ; A61K31/4196 ; A61P19/00 ; C07D401/14 ; C07D403/14
摘要：
N 3 -Heteroaryl substituted triazoles and N 5 -heteroaryl substituted triazoles and pharmaceutical compositions containing the compounds are disclosed as being useful in inhibiting the activity of the receptor protein tyrosine kinase Axl. Methods of using the compounds in treating diseases or conditions associated with Axl activity are also disclosed.
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