发明公开
- 专利标题: SEROTONIN REUPTAKE INHIBITORS
- 专利标题(中): 选择性五羟色胺再摄取抑制剂
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申请号: EP11773367.5申请日: 2011-10-10
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公开(公告)号: EP2627630A1公开(公告)日: 2013-08-21
- 发明人: STANGELAND, Eric L. , PATTERSON, Lori Jean , SAITO, Daisuke Roland
- 申请人: Theravance, Inc.
- 申请人地址: 901 Gateway Boulevard South San Francisco, CA 94080 US
- 专利权人: Theravance, Inc.
- 当前专利权人: Theravance, Inc.
- 当前专利权人地址: 901 Gateway Boulevard South San Francisco, CA 94080 US
- 代理机构: Scott, Susan Margaret
- 优先权: US391758P 20101011
- 国际公布: WO2012051103 20120419
- 主分类号: C07D207/08
- IPC分类号: C07D207/08 ; C07D401/12 ; A61K31/40 ; A61P11/00
摘要:
In one aspect, the invention relates to compounds of formula I: (I) where X, Y, R
1 , R
2 , R
3 , R
4 , R
4 , and n are as defined in the specification, or a pharmaceutically acceptable salt thereof. The compounds of formula I are serotonin reuptake inhibitors. In another aspect, the invention relates to pharmaceutical compositions comprising such compounds; methods of using such compounds; and process and intermediates for preparing such compounds.
1 , R
2 , R
3 , R
4 , R
4 , and n are as defined in the specification, or a pharmaceutically acceptable salt thereof. The compounds of formula I are serotonin reuptake inhibitors. In another aspect, the invention relates to pharmaceutical compositions comprising such compounds; methods of using such compounds; and process and intermediates for preparing such compounds.
公开/授权文献
- EP2627630B1 SEROTONIN REUPTAKE INHIBITORS 公开/授权日:2014-12-31
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