发明申请
US20050020576A1 Kappa agonist compounds and pharmaceutical formulations thereof
审中-公开
卡帕激动剂化合物及其药物制剂
- 专利标题： Kappa agonist compounds and pharmaceutical formulations thereof
- 专利标题（中）： 卡帕激动剂化合物及其药物制剂
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申请号： US10807113申请日： 2004-03-23
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公开(公告)号： US20050020576A1公开(公告)日： 2005-01-27
- 发明人: Wei Zhang , Alan Maycock , Michael Marella , Virendra Kumar , Forrest Gaul , Michael Chang , Deqi Guo
- 申请人： Wei Zhang , Alan Maycock , Michael Marella , Virendra Kumar , Forrest Gaul , Michael Chang , Deqi Guo
- 专利权人： Adolor Corporation
- 当前专利权人： Adolor Corporation
- 主分类号： A61K31/404
- IPC分类号： A61K31/404 ; A61K31/4439 ; A61K45/06 ; C07D207/12 ; C07D209/42 ; C07D213/56 ; C07D241/04 ; C07D295/073 ; C07D403/06 ; A61K31/55 ; A61K31/40 ; A61K31/445
摘要：
Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics are provided. The compounds of formulae I, II, IIA, III, IIIA, IIIB, IIB-i, IV and IVA have the structure: wherein R1, R2, R3, R4; and X, X4, X5, X7, X9; Y, Z and n are as described in the specification.
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