发明申请
- 专利标题： Substituted diketopiperazines as oxytocin antagonists
- 专利标题（中）： 取代的二酮哌嗪作为催产素拮抗剂
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申请号： US10499177申请日： 2002-12-20
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公开(公告)号： US20050148572A1公开(公告)日： 2005-07-07
- 发明人: Alan Borthwick , Richard Hatley , Deirdre Hickey , John Liddle , David Livermore , Andrew Mason , Neil Miller , Fabrizio Nerozzi , Steven Sollis , Anna Szardenings , Paul Wyatt
- 申请人： Alan Borthwick , Richard Hatley , Deirdre Hickey , John Liddle , David Livermore , Andrew Mason , Neil Miller , Fabrizio Nerozzi , Steven Sollis , Anna Szardenings , Paul Wyatt
- 优先权： GB0130677.8 20011221
- 国际申请： PCT/EP02/14823 WO 20021220
- 主分类号： C07D241/04
- IPC分类号： C07D241/04 ; A61K31/495 ; A61K31/496 ; A61K31/5377 ; A61K31/541 ; A61K31/551 ; A61K38/00 ; A61P15/06 ; A61P43/00 ; C07D401/06 ; C07D401/12 ; C07D403/06 ; C07D403/10 ; C07D417/12 ; C07D491/113 ; C07K5/06 ; C07K5/065 ; C07D413/02 ; C07D43/02
摘要：
A method of treating or preventing diseases or conditions mediated through the action of oxytocin which comprises administering to a mammal in need thereof of an effective amount of a compound of the formula (I) and/or a physiologically acceptable derivative thereof, wherein the substituents have the meaning given in the description. Disclosed are also novel compounds of formula (I) and processes for their preparation.
公开/授权文献
- US07514437B2 Substituted diketopiperazines as oxytocin antagonists 公开/授权日：2009-04-07