发明申请
- 专利标题： Process for the Preparation of Gabapentin
- 专利标题（中）： 加巴喷丁的制备方法
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申请号： US11571192申请日： 2005-06-22
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公开(公告)号： US20080097122A1公开(公告)日： 2008-04-24
- 发明人: Marco Villa , Maurizio Paiocchi , Katiuscia Arrighi , Francesco Corcella , Vincenzo Cannata , Giorgio Soriato , Massimo Verzini
- 申请人： Marco Villa , Maurizio Paiocchi , Katiuscia Arrighi , Francesco Corcella , Vincenzo Cannata , Giorgio Soriato , Massimo Verzini
- 申请人地址： IT Bresso (Milan) Italy
- 专利权人： AAMBON GROUPS P.P.A.
- 当前专利权人： AAMBON GROUPS P.P.A.
- 当前专利权人地址： IT Bresso (Milan) Italy
- 优先权： ITM12004A001271 20040624
- 国际申请： PCT/EP05/52906 WO 20050622
- 主分类号： C07C231/10
- IPC分类号： C07C231/10
摘要：
The present invention relates to a process for the preparation of gabapentin and, more in particular, to a method of synthesis of 1,1-cyclohexane acetic acid monoamide, an intermediate used in the preparation of gabapentin, comprising the basic hydrolysis reaction of α,−-diaminocarbonyl-β,β-pentamethylene glutarimide.
公开/授权文献
- US07759517B2 Process for the preparation of gabapentin 公开/授权日：2010-07-20