发明申请
US20090318702A1 PROCESS FOR PRODUCTION OF 4-OXOQUINOLINE COMPOUND 有权
4-氧杂环戊烯化合物的生产方法

PROCESS FOR PRODUCTION OF 4-OXOQUINOLINE COMPOUND
摘要:
The present invention provides a compound useful as a synthetic intermediate for an anti-HIV agent having an integrase inhibitory activity, a production method thereof, and a production method of an anti-HIV agent using the synthetic intermediate. Specifically, the present invention provides, for example, compounds represented by the formulas (6), (7-1), (7-2) and (8): wherein R is a fluorine atom or a methoxy group, R1 is a C1-C4 alkyl group, R2 is a hydroxyl-protecting group, and X2 is a halogen atom, a production method thereof, and a production method of an anti-HIV agent using the synthetic intermediate.
公开/授权文献
信息查询
0/0