发明申请
US20100004208A1 SUBSTITUTED BENZOFURANS, BENZOTHIOPHENES, BENZOSELENOPHENES AND INDOLES AND THEIR USE AS TUBULIN POLYMERISATION INHIBITORS
有权
替代苯唑酮,苯并噻唑,苯并噻吩和吲哚,以及其作为管状体聚合抑制剂的用途
- 专利标题: SUBSTITUTED BENZOFURANS, BENZOTHIOPHENES, BENZOSELENOPHENES AND INDOLES AND THEIR USE AS TUBULIN POLYMERISATION INHIBITORS
- 专利标题(中): 替代苯唑酮,苯并噻唑,苯并噻吩和吲哚,以及其作为管状体聚合抑制剂的用途
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申请号: US12162917申请日: 2007-02-02
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公开(公告)号: US20100004208A1公开(公告)日: 2010-01-07
- 发明人: Jason Hugh Chaplin , Gurmit Singh Gill , Damian Wojciech Grobelny , Bernard Luke Flynn , Gabriel Kremmidiotis
- 申请人: Jason Hugh Chaplin , Gurmit Singh Gill , Damian Wojciech Grobelny , Bernard Luke Flynn , Gabriel Kremmidiotis
- 申请人地址: AU Thebarton
- 专利权人: BIONOMICS LIMITED
- 当前专利权人: BIONOMICS LIMITED
- 当前专利权人地址: AU Thebarton
- 国际申请: PCT/AU2007/000101 WO 20070202
- 主分类号: A61K31/343
- IPC分类号: A61K31/343 ; C07D307/78 ; C07D307/82 ; C07D405/12 ; A61K31/443 ; A61K31/496 ; A61K31/665 ; A61P35/00
摘要:
The present invention relates generally to substituted benzofurans, benzothiophenes, and indoles and their use as tubulin polymerisation inhibitors.