Invention Application
US20110212945A1 AZABIPHENYLAMINOBENZOIC ACID DERIVATIVES AS DHODH INHIBITORS
失效
作为DHODH抑制剂的亚氨基苯甲酸苯甲酸衍生物
- Patent Title: AZABIPHENYLAMINOBENZOIC ACID DERIVATIVES AS DHODH INHIBITORS
- Patent Title (中): 作为DHODH抑制剂的亚氨基苯甲酸苯甲酸衍生物
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Application No.: US12672725Application Date: 2008-08-08
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Publication No.: US20110212945A1Publication Date: 2011-09-01
- Inventor: Julio Cesar Castro Palomino Laria , Emma Terricabras Belart , Montserrat Erra Sola , Eloisa Navarro Romero , Silvia Fonquerna Pou , Aranzazu Cardus Figueras , Maria Estrella Lozoya Toribio
- Applicant: Julio Cesar Castro Palomino Laria , Emma Terricabras Belart , Montserrat Erra Sola , Eloisa Navarro Romero , Silvia Fonquerna Pou , Aranzazu Cardus Figueras , Maria Estrella Lozoya Toribio
- Applicant Address: ES Barcelona
- Assignee: ALMIRALL, S.A.
- Current Assignee: ALMIRALL, S.A.
- Current Assignee Address: ES Barcelona
- Priority: ESP200702261 20070810; EP08382011.8 20080313
- International Application: PCT/EP2008/006573 WO 20080808
- Main IPC: A61K31/55
- IPC: A61K31/55 ; C07D213/74 ; A61K31/4418 ; C07D401/04 ; A61K31/506 ; C07D413/10 ; A61K31/4439 ; C07D239/42 ; A61K31/505 ; A61K31/444 ; C07D401/10 ; A61K31/4709 ; A61K31/4545 ; C07D413/04 ; A61K31/5377 ; A61P19/00 ; A61P29/00 ; A61P35/00 ; A61P31/12 ; A61P31/00

Abstract:
The present disclosure relates to new azabiphenylaminobenzoic acid derivatives of formula (I); as well as processes for their preparation, pharmaceutical compositions comprising them, and their use in therapy as inhibitors of the dehydroorotate dihydrogenase (DHODH).
Public/Granted literature
- US08536165B2 Azabiphenylaminobenzoic acid derivatives as DHODH inhibitors Public/Granted day:2013-09-17
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