发明申请
- 专利标题： TRIAZOLOPYRIDINES
- 专利标题（中）： 三唑并[
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申请号： US13512701申请日： 2010-11-17
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公开(公告)号： US20120328610A1公开(公告)日： 2012-12-27
- 发明人: Volker Schulze , Marcus Koppitz , Dirk Kosemund , Hartmut Schirok , Benjamin Bader , Philip Lienau , Antje Margret Wengner , Hans Briem , Simon Holton , Gerhard Siemeister , Stefan Prechtl , Ulf Bömer
- 申请人： Volker Schulze , Marcus Koppitz , Dirk Kosemund , Hartmut Schirok , Benjamin Bader , Philip Lienau , Antje Margret Wengner , Hans Briem , Simon Holton , Gerhard Siemeister , Stefan Prechtl , Ulf Bömer
- 申请人地址： DE Monheim
- 专利权人： BAYER INTELLECTUAL PROPERTY GMBH
- 当前专利权人： BAYER INTELLECTUAL PROPERTY GMBH
- 当前专利权人地址： DE Monheim
- 优先权： EP09075535.6 20091130
- 国际申请： PCT/EP2010/006994 WO 20101117
- 主分类号： A61K31/437
- IPC分类号： A61K31/437 ; A61K31/444 ; A61K31/496 ; A61K31/5377 ; A61K31/4545 ; A61K31/573 ; A61K31/567 ; A61K31/4745 ; A61K31/704 ; A61K38/14 ; A61K31/664 ; A61K31/513 ; A61K31/7076 ; A61K31/69 ; A61K33/24 ; A61K31/519 ; A61K39/395 ; A61P35/00 ; A61P35/02 ; A61P35/04 ; A61K31/7068 ; A61K31/52 ; C07D471/04
摘要：
The present invention relates to triazolopyridine compounds of general formula (I) which are Monopolar Spindle 1 kinase (Mps-1 or TTK) inhibitors: Formula (I), in which R1, R2, R3, R4, and R5 are as given in the description and in the claims, to methods of preparing said compounds, to pharmaceutical compositions and combinations comprising said compounds, to the use of said compounds for manufacturing a pharmaceutical composition for the treatment or prophylaxis proliferative of diseases, as well as to intermediate compounds useful in the preparation of said compounds.
公开/授权文献
- US09676766B2 Triazolopyridines 公开/授权日：2017-06-13
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