发明申请
- 专利标题： CARRIER LINKED PALIPERIDONE PRODRUGS
- 专利标题（中）： CARRIER连接的PALIPERIDONE PRODRUGS
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申请号： US13500611申请日： 2010-10-06
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公开(公告)号： US20130053405A1公开(公告)日： 2013-02-28
- 发明人: Ulrich Hersel , Harald Rau , Guillaume Maitro , Thomas Wegge
- 申请人： Ulrich Hersel , Harald Rau , Guillaume Maitro , Thomas Wegge
- 优先权： EP09172334.6 20091006; EP09180531.7 20091223; EP10171511.8 20100730
- 国际申请： PCT/EP2010/064874 WO 20101006
- 主分类号： C07D413/14
- IPC分类号： C07D413/14 ; A61P25/00 ; A61P25/24 ; A61K31/519 ; A61P25/18
摘要：
The present invention relates to prodrugs or a pharmaceutically acceptable salt thereof comprising a covalent Paliperidone carrier conjugate of formula (I) wherein Z0 is defined in the description and the claims as well as pharmaceutical composition comprising said compounds. The compounds are useful as medicament, especially for diseases or disorders which can be treated by Paliperidone.
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