发明申请
- 专利标题: CEPHEM COMPOUND HAVING CATECHOL GROUP
- 专利标题(中): CEPHEM化合物有CATECHOL集团
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申请号: US13639412申请日: 2011-04-04
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公开(公告)号: US20130102583A1公开(公告)日: 2013-04-25
- 发明人: Shinya Hisakawa , Yasushi Hasegawa , Toshiaki Aoki , Hiroki Kusano , Masayuki Sano , Jun Sato , Kenji Yamawaki
- 申请人: Shinya Hisakawa , Yasushi Hasegawa , Toshiaki Aoki , Hiroki Kusano , Masayuki Sano , Jun Sato , Kenji Yamawaki
- 申请人地址: JP Osaka-shi, Osaka
- 专利权人: SHIONOGI & CO., LTD.
- 当前专利权人: SHIONOGI & CO., LTD.
- 当前专利权人地址: JP Osaka-shi, Osaka
- 优先权: JP2010-087131 20100405; JP2010-274180 20101209
- 国际申请: PCT/JP2011/058498 WO 20110404
- 主分类号: C07D505/24
- IPC分类号: C07D505/24 ; C07D471/08 ; C07D501/56
摘要:
A compound of the formula: wherein X is —N═, —CH═, or the like; W is —CH2— or the like; U is —S— or the like; R1 and R2 are each independently hydrogen, halogen, optionally substituted lower alkyl, or the like; R3 is hydrogen or the like; each R4 is independently hydrogen, halogen, or the like; m is an integer from 0 to 2; Q is a single bond, or the like; G is —C(═O)—, or the like; D is a single bond, —NH—, or the like; and E is a cyclic quaternary ammonium group, or an ester, a protected compound at the amino on the ring in the 7-side chain, a pharmaceutically acceptable salt, or a solvate thereof.
公开/授权文献
- US09145425B2 Cephem compound having catechol group 公开/授权日:2015-09-29