Invention Application
US20160355536A1 METHOD FOR PRODUCING THIOLANE SKELETON-TYPE GLYCOCONJUGATE, AND THIOLANE SKELETON-TYPE GLYCOCONJUGATE
有权
用于生产硫醇酮型糖苷酸盐的方法,以及硫醇型骨架型糖蛋白
- Patent Title: METHOD FOR PRODUCING THIOLANE SKELETON-TYPE GLYCOCONJUGATE, AND THIOLANE SKELETON-TYPE GLYCOCONJUGATE
- Patent Title (中): 用于生产硫醇酮型糖苷酸盐的方法,以及硫醇型骨架型糖蛋白
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Application No.: US15238232Application Date: 2016-08-16
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Publication No.: US20160355536A1Publication Date: 2016-12-08
- Inventor: Takayuki ITO , Toru WATANABE , Hideki OKADA , Hidenobu KUNIYOSHI
- Applicant: FUJIFILM Corporation
- Applicant Address: JP Tokyo
- Assignee: FUJIFILM Corporation
- Current Assignee: FUJIFILM Corporation
- Current Assignee Address: JP Tokyo
- Priority: JP2014-029020 20140218; JP2014-220368 20141029
- Main IPC: C07H13/08
- IPC: C07H13/08 ; C07D333/32 ; C07H15/04

Abstract:
There is provided a production method of a compound represented by the following formula (II) through a step of reacting a compound represented by the following General Formula (I) with a sulfur compound. In General Formulas (I) and (II), R1 represents a hydrogen atom or an acyl group, R2 represents a hydrogen atom, a fluorine atom, an acyloxy group, an arylmethyloxy group, an allyloxy group, an arylmethyloxycarbonyloxy group, or an allyloxycarbonyloxy group, R3 represents a hydrogen atom or an acyloxy group, R5 represents an alkyl group or an aryl group, and X represents a leaving group. Here, in a case where R2 is a fluorine atom, an acyloxy group, an arylmethyloxy group, an allyloxy group, an arylmethyloxycarbonyloxy group, or an allyloxycarbonyloxy group, R3 is an acyloxy group.
Public/Granted literature
- US09884882B2 Method for producing thiolane skeleton-type glycoconjugate, and thiolane skeleton-type glycoconjugate Public/Granted day:2018-02-06
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