发明授权
US5723483A Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensin
receptors, their preparation and pharmaceutical compositions containing
them
失效
对神经降压素受体有活性的取代的1-苯基-3-吡唑酰胺，其制剂和含有它们的药物组合物
- 专利标题： Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensin receptors, their preparation and pharmaceutical compositions containing them
- 专利标题（中）： 对神经降压素受体有活性的取代的1-苯基-3-吡唑酰胺，其制剂和含有它们的药物组合物
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申请号： US630761申请日： 1996-04-10
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公开(公告)号： US5723483A公开(公告)日： 1998-03-03
- 发明人: Bernard Labeeuw , Danielle Gully , Francis Jeanjean , Jean-Charles Molimard , Robert Boigegrain
- 申请人： Bernard Labeeuw , Danielle Gully , Francis Jeanjean , Jean-Charles Molimard , Robert Boigegrain
- 申请人地址： FRX Paris
- 专利权人： Sanofi
- 当前专利权人： Sanofi
- 当前专利权人地址： FRX Paris
- 优先权： FRX9404350 19950411
- 主分类号： A61K31/415
- IPC分类号： A61K31/415 ; A61K31/4155 ; A61K31/42 ; A61K31/435 ; A61K31/439 ; A61K31/44 ; A61K31/4427 ; A61K31/4439 ; A61K31/445 ; A61K31/454 ; A61K31/495 ; A61K31/496 ; A61K31/535 ; A61K31/5377 ; A61P1/00 ; A61P25/00 ; A61P35/00 ; A61P43/00 ; C07C61/20 ; C07C62/34 ; C07C243/22 ; C07C255/66 ; C07C309/45 ; C07C309/47 ; C07C311/21 ; C07D231/12 ; C07D231/14 ; C07D231/38 ; C07D233/62 ; C07D401/10 ; C07D401/12 ; C07D403/10 ; C07D403/12 ; C07D413/04 ; C07D413/12 ; C07D453/02 ; A01N43/56
摘要：
The invention relates to new substituted 1-phenyl-3-pyrazolecarboxamides having a great affinity for human neurotensin receptors, to a process for preparing them and to pharmaceutical compositions containing them as active principles. More particularly, this invention relates to the discovery that the affinity for neurotensin receptors, especially human neurotensin receptors, is increased by substituting the phenyl group of 1-phenyl-3-pyrazolecarboxamide compounds with particular groups.
公开/授权文献
- US5136431A Zoom lens of the internal focus type 公开/授权日：1992-08-04
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