发明授权
- 专利标题: Erythromycin a derivatives and method for preparing same
- 专利标题(中): 红霉素a衍生物及其制备方法
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申请号: US07869111申请日: 1992-04-14
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公开(公告)号: US06342590B1公开(公告)日: 2002-01-29
- 发明人: Shigeo Morimoto , Takashi Adachi , Tohru Matsunaga , Masato Kashimura , Yoshiaki Watanabe , Kaoru Sota
- 申请人: Shigeo Morimoto , Takashi Adachi , Tohru Matsunaga , Masato Kashimura , Yoshiaki Watanabe , Kaoru Sota
- 优先权: JP2-220315 19860918
- 主分类号: C07H100
- IPC分类号: C07H100
摘要:
Erythromycin A derivatives represented by the general formula wherein R1 is a 2-alkenyl group having 3 to 15 carbon atoms, an arylmethyl group, or an arylmethyl group substituted by 1 to 3 of a halogen atom, an alkoxy group 1 to 4 carbon atoms, a nitro group or an alkoxycarbonyl group having 2 to 6 carbon atoms, R2 is a substituted silyl group and R3 is a hydrogen atom or R2, are disclosed. These compounds are useful as intermediates of the anti-bacterial agents.