Invention Grant
- Patent Title: Guanidine mimics as factor Xa inhibitors
- Patent Title (中): 胍类似物作为因子Xa抑制剂
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Application No.: US11197978Application Date: 2005-08-05
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Publication No.: US07235575B2Publication Date: 2007-06-26
- Inventor: Patrick Y. Lam , Charles G. Clark , Celia Dominguez , John M. Fevig , Qi Han , Renhua Li , Donald J P Pinto , James R. Pruitt , Mimi L. Quan
- Applicant: Patrick Y. Lam , Charles G. Clark , Celia Dominguez , John M. Fevig , Qi Han , Renhua Li , Donald J P Pinto , James R. Pruitt , Mimi L. Quan
- Applicant Address: US NJ Princeton
- Assignee: Bristol Myers Squibb Company
- Current Assignee: Bristol Myers Squibb Company
- Current Assignee Address: US NJ Princeton
- Agent Jing G. Sun; David H. Vance
- Main IPC: A61K31/423
- IPC: A61K31/423 ; C07D413/04 ; A61K31/44 ; C07D471/02 ; C07D491/02

Abstract:
The present application describes nitrogen containing heteroaromatics and derivatives thereof of formula I: or pharmaceutically acceptable salt forms thereof, wherein rings D-E represent guanidine mimics, which are useful as inhibitors of factor Xa.
Public/Granted literature
- US20060040973A1 Novel guanidine mimics as factor Xa inhibitors Public/Granted day:2006-02-23
Information query
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