Invention Grant
- Patent Title: Nitrogen-containing aromatic derivatives
- Patent Title (中): 含氮芳香族衍生物
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Application No.: US10420466Application Date: 2003-04-18
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Publication No.: US07253286B2Publication Date: 2007-08-07
- Inventor: Yasuhiro Funahashi , Akihiko Tsuruoka , Masayuki Matsukura , Toru Haneda , Yoshio Fukuda , Junichi Kamata , Keiko Takahashi , Tomohiro Matsushima , Kazuki Miyazaki , Ken-ichi Nomoto , Tatsuo Watanabe , Hiroshi Obaishi , Atsumi Yamaguchi , Sachi Suzuki , Katsuji Nakamura , Fusayo Mimura , Yuji Yamamoto , Junji Matsui , Kenji Matsui , Takako Yoshiba , Yasuyuki Suzuki , Itaru Arimoto
- Applicant: Yasuhiro Funahashi , Akihiko Tsuruoka , Masayuki Matsukura , Toru Haneda , Yoshio Fukuda , Junichi Kamata , Keiko Takahashi , Tomohiro Matsushima , Kazuki Miyazaki , Ken-ichi Nomoto , Tatsuo Watanabe , Hiroshi Obaishi , Atsumi Yamaguchi , Sachi Suzuki , Katsuji Nakamura , Fusayo Mimura , Yuji Yamamoto , Junji Matsui , Kenji Matsui , Takako Yoshiba , Yasuyuki Suzuki , Itaru Arimoto
- Applicant Address: JP Bunkyo-ku, Tokyo
- Assignee: Eisai Co., Ltd
- Current Assignee: Eisai Co., Ltd
- Current Assignee Address: JP Bunkyo-ku, Tokyo
- Agency: Choate, Hall & Stewart LLP
- Agent Andrea L. C. Robidoux
- Priority: JPP2000-320420 20001020; JPP2000-386195 20001220; JPP2001-046685 20010222
- Main IPC: A61K31/47
- IPC: A61K31/47 ; C07D215/16

Abstract:
Compounds represented by the following general formula: [wherein Ag is an optionally substituted 5- to 14-membered heterocyclic group, etc.; Xg is —O—, —S—, etc.; Yg is an optionally substituted C6-14 aryl group, an optionally substituted 5- to 14-membered heterocyclic group, etc.; and Tg1 is a group represented by the following general formula: (wherein Eg is a single bond or —N(Rg2)—, Rg1 and Rg2 each independently represent a hydrogen atom, an optionally substituted C1-6 alkyl group, etc. and Zg represents a C1-8 alkyl group, a C3-8 alicyclic hydrocarbon group, a C6-14 aryl group, etc.)], salts thereof or hydrates of the foregoing.
Public/Granted literature
- US20040053908A1 Nitrogen-containing aromatic derivatives Public/Granted day:2004-03-18
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