发明授权
- 专利标题: Phenoxy-substituted pyrimidines as opioid receptor modulators
- 专利标题(中): 苯氧基取代的嘧啶作为阿片受体调节剂
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申请号: US12913948申请日: 2010-10-28
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公开(公告)号: US08394809B2公开(公告)日: 2013-03-12
- 发明人: Steven J. Coats , Yue-Mei Zhang , Shu-Chen Lin , Li Liu , Tamara A. Miskowski , Scott L. Dax , Henry Breslin , Bart L. De Corte , Wei He
- 申请人: Steven J. Coats , Yue-Mei Zhang , Shu-Chen Lin , Li Liu , Tamara A. Miskowski , Scott L. Dax , Henry Breslin , Bart L. De Corte , Wei He
- 申请人地址: BE
- 专利权人: Janssen Pharmaceutica, NV
- 当前专利权人: Janssen Pharmaceutica, NV
- 当前专利权人地址: BE
- 主分类号: A01N43/54
- IPC分类号: A01N43/54 ; A61K31/505
摘要:
Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula I as follows: wherein R1, Y, R2, R3, and Ra are defined herein.