-
公开(公告)号:US08394809B2
公开(公告)日:2013-03-12
申请号:US12913948
申请日:2010-10-28
申请人: Steven J. Coats , Yue-Mei Zhang , Shu-Chen Lin , Li Liu , Tamara A. Miskowski , Scott L. Dax , Henry Breslin , Bart L. De Corte , Wei He
发明人: Steven J. Coats , Yue-Mei Zhang , Shu-Chen Lin , Li Liu , Tamara A. Miskowski , Scott L. Dax , Henry Breslin , Bart L. De Corte , Wei He
IPC分类号: A01N43/54 , A61K31/505
CPC分类号: C07D239/52 , A61K31/506 , C07D239/28 , C07D239/34 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/12
摘要: Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula I as follows: wherein R1, Y, R2, R3, and Ra are defined herein.
摘要翻译: 公开了用于治疗各种疾病,综合征,病症和障碍(包括疼痛)的化合物,组合物和方法。 这样的化合物由式I表示如下:其中R1,Y,R2,R3和Ra在本文中定义。
-
公开(公告)号:US20110105455A1
公开(公告)日:2011-05-05
申请号:US12913948
申请日:2010-10-28
申请人: STEVEN J. COATS , Yue-Mei Zhang , Shu-Chen Lin , Li Liu , Tamara A. Miskowski , Scott L. Dax , Henry Breslin , Bart L. De Corte , Wei He
发明人: STEVEN J. COATS , Yue-Mei Zhang , Shu-Chen Lin , Li Liu , Tamara A. Miskowski , Scott L. Dax , Henry Breslin , Bart L. De Corte , Wei He
IPC分类号: A61K31/506 , C07D403/12 , C07D401/12 , C07D413/12 , C07D417/12 , C07D401/14 , A61K31/505 , A61K31/5377 , A61P29/00 , A61P25/04 , A61P25/16 , A61P25/30 , A61P25/32 , A61P1/12 , A61P9/00 , A61P15/00 , A61P11/00
CPC分类号: C07D239/52 , A61K31/506 , C07D239/28 , C07D239/34 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/12
摘要: Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula I as follows: wherein R1, Y, R2, R3, and Ra are defined herein.
摘要翻译: 公开了用于治疗各种疾病,综合征,病症和障碍(包括疼痛)的化合物,组合物和方法。 这样的化合物由式I表示如下:其中R1,Y,R2,R3和Ra在本文中定义。
-
公开(公告)号:US08513271B2
公开(公告)日:2013-08-20
申请号:US12913966
申请日:2010-10-28
申请人: Steven J. Coats , Haiyan Bian , Peter J. Connolly , Gilles Bignan , Chaozhong Cai , Scott L. Dax , Bart L. DeCorte , Shu-Chen Lin , Li Liu , Mark J. Macielag , Philip M. Pitis , Yue-Mei Zhang , Bin Zhu , Wei He
发明人: Steven J. Coats , Haiyan Bian , Peter J. Connolly , Gilles Bignan , Chaozhong Cai , Scott L. Dax , Bart L. DeCorte , Shu-Chen Lin , Li Liu , Mark J. Macielag , Philip M. Pitis , Yue-Mei Zhang , Bin Zhu , Wei He
IPC分类号: A01N43/54
CPC分类号: C07D239/47 , C07D401/04 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14
摘要: Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula I as follows: wherein R1, R2, R3, and L, A, and Ra are defined herein.
摘要翻译: 公开了用于治疗各种疾病,综合征,病症和障碍(包括疼痛)的化合物,组合物和方法。 这样的化合物由式I表示如下:其中R1,R2,R3和L,A和Ra在本文中定义。
-
4.4-SUBSTITUTED-2-PHENOXY-PHENYLAMINE DELTA OPIOID RECEPTOR MODULATORS 有权
标题翻译: 4-取代-2-苯基 - 苯甲酰三嗪类阿片受体调节剂公开(公告)号:US20120302541A1
公开(公告)日:2012-11-29
申请号:US13503433
申请日:2010-10-28
申请人: Steven J. Coats , Haiyan Bian , Chaozhong Cai , Bart L. DeCorte , Li Liu , Mark J. Macielag , Scott L. Dax , Philip M. Pitis , Peter J. Connolly , Wei He
发明人: Steven J. Coats , Haiyan Bian , Chaozhong Cai , Bart L. DeCorte , Li Liu , Mark J. Macielag , Scott L. Dax , Philip M. Pitis , Peter J. Connolly , Wei He
IPC分类号: A61K31/40 , C07D211/26 , A61K31/445 , C07D401/12 , A61K31/4439 , C07D405/12 , A61K31/4025 , C07D409/12 , C07D403/12 , A61K31/506 , C07D295/096 , A61K31/495 , C07D413/12 , A61K31/4245 , C07D451/02 , A61K31/46 , C07C217/84 , A61K31/136 , C07D205/04 , A61K31/397 , C07D453/02 , A61K31/439 , A61P29/00 , A61P19/02 , A61P25/06 , A61P11/02 , A61P13/10 , A61P17/00 , A61P11/12 , A61P25/00 , A61P25/02 , A61P1/00 , A61P35/00 , A61P25/24 , A61P25/16 , A61P25/30 , A61P25/32 , A61P13/00 , A61P15/00 , A61P1/12 , A61P9/00 , A61P11/00 , C07D207/14
CPC分类号: C07D401/12 , C07C211/48 , C07C211/50 , C07C233/08 , C07C233/11 , C07C233/65 , C07C255/50 , C07D205/04 , C07D207/09 , C07D211/56 , C07D405/12 , C07D409/12 , C07D413/12 , C07D451/04 , C07D453/02
摘要: Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula I as follows: wherein R1, R2, R3, Ra, and Y are defined herein.
摘要翻译: 公开了用于治疗各种疾病,综合征,病症和障碍(包括疼痛)的化合物,组合物和方法。 这样的化合物由式I表示如下:其中R1,R2,R3,Ra和Y如本文所定义。
-
5.4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators 有权
标题翻译: 4-取代-2-苯氧基 - 苯胺δ阿片样物质受体调节剂公开(公告)号:US08846655B2
公开(公告)日:2014-09-30
申请号:US13503433
申请日:2010-10-28
申请人: Steven J. Coats , Haiyan Bian , Chaozhong Cai , Bart L. DeCorte , Li Liu , Mark J. Macielag , Scott L. Dax , Philip M. Pitis , Peter J. Connolly , Wei He
发明人: Steven J. Coats , Haiyan Bian , Chaozhong Cai , Bart L. DeCorte , Li Liu , Mark J. Macielag , Scott L. Dax , Philip M. Pitis , Peter J. Connolly , Wei He
IPC分类号: A61K31/40 , A61K31/445 , A61K31/4439 , A61K31/4025 , A61K31/506 , A61K31/495 , C07D211/56 , C07D405/12 , C07D207/09 , C07C255/50 , C07C211/48 , C07D413/12 , C07D401/12 , C07C211/50 , C07D205/04 , C07C233/08 , C07C233/11 , C07C233/65 , C07D451/04 , C07D453/02 , C07D409/12
CPC分类号: C07D401/12 , C07C211/48 , C07C211/50 , C07C233/08 , C07C233/11 , C07C233/65 , C07C255/50 , C07D205/04 , C07D207/09 , C07D211/56 , C07D405/12 , C07D409/12 , C07D413/12 , C07D451/04 , C07D453/02
摘要: Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula I as follows: wherein R1, R2, R3, Ra, and Y are defined herein.
摘要翻译: 公开了用于治疗各种疾病,综合征,病症和障碍(包括疼痛)的化合物,组合物和方法。 这样的化合物由式I表示如下:其中R1,R2,R3,Ra和Y如本文所定义。
-
公开(公告)号:US08324380B2
公开(公告)日:2012-12-04
申请号:US12256891
申请日:2008-10-23
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: C07D251/30 , C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D401/12 , C07D403/12 , A61K31/53 , A61P1/12 , A61P1/06 , A61P1/00
CPC分类号: C07D251/38 , C07D401/12 , C07D403/12 , C07D405/14
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
-
公开(公告)号:US20140038968A1
公开(公告)日:2014-02-06
申请号:US13653452
申请日:2012-10-17
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: C07D251/38 , C07D403/12
CPC分类号: C07D251/38 , C07D401/12 , C07D403/12 , C07D405/14
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
-
公开(公告)号:US08362247B2
公开(公告)日:2013-01-29
申请号:US13113751
申请日:2011-05-23
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: C07D403/06 , C07D403/12 , C07D403/14 , C07D401/06 , C07D401/12 , C07D401/14 , A61K31/506 , A61P1/00 , A61P1/06
CPC分类号: C07D239/545 , C07D251/20 , C07D251/34 , C07D251/38 , C07D251/46 , C07D403/12
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体及其衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
-
公开(公告)号:US07968710B2
公开(公告)日:2011-06-28
申请号:US11375407
申请日:2006-03-14
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: C07D251/30 , C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D401/12 , C07D403/12 , A61K31/53 , A61P1/12 , A61P1/06 , A61P1/00
CPC分类号: C07D239/545 , C07D251/20 , C07D251/34 , C07D251/38 , C07D251/46 , C07D403/12
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
-
公开(公告)号:US20120129862A1
公开(公告)日:2012-05-24
申请号:US13113751
申请日:2011-05-23
申请人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
发明人: Steven J. Coats , Alexey B. Dyatkin , Wei He , Joseph Lisko , Tamara A. Miskowski , Janet L. Ralbovsky , Mark J. Schulz
IPC分类号: A61K31/53 , C07D403/12 , C07D251/20 , A61P29/00 , C07D251/38 , A61P1/00 , A61P1/12 , A61P35/00 , C07D251/46 , C07D251/30
CPC分类号: C07D239/545 , C07D251/20 , C07D251/34 , C07D251/38 , C07D251/46 , C07D403/12
摘要: The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1 receptor mediated disorders.
摘要翻译: 本发明涉及某些新的式(I)化合物:以及制备这些化合物,组合物,中间体和衍生物以及用于治疗促动蛋白原1或原激素1受体介导的病症的方法。
-
-
-
-
-
-
-
-
-