Invention Grant
- Patent Title: Anti-aging agent containing arctigenin derivative
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Application No.: US14389200Application Date: 2013-03-27
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Publication No.: US09675538B2Publication Date: 2017-06-13
- Inventor: Yuya Hayashi , Yoko Mizutare
- Applicant: ROHTO Pharmaceutical Co., Ltd.
- Applicant Address: JP Osaka
- Assignee: Rohto Pharmaceutical Co., Ltd.
- Current Assignee: Rohto Pharmaceutical Co., Ltd.
- Current Assignee Address: JP Osaka
- Agency: Knobbe, Martens, Olson & Bear, LLP
- Priority: JP2012-081177 20120330
- International Application: PCT/JP2013/059128 WO 20130327
- International Announcement: WO2013/146943 WO 20131003
- Main IPC: A61K8/00
- IPC: A61K8/00 ; A61K8/49 ; A61Q19/02 ; A61Q19/08 ; A61K31/365 ; C07D307/33

Abstract:
An arctigenin derivative used for anti-aging treatment, including protection of the skin from the sun and recovery of skin elasticity. A variety of fatty acid ester derivatives, alcohol ether derivatives and alkylated derivatives are used as the arctigenin derivatives. Agents for controlling ET-1 production, elastase inhibitors, and anti-inflammatory agents are prepared. Such arctigenin derivatives are particularly useful as an external agent for the skin, such as an anti-inflammatory external agent, a sunscreen external agent, or an external agent for recovering elasticity.
Public/Granted literature
- US20150093345A1 ANTI-AGING AGENT CONTAINING ARCTIGENIN DERIVATIVE Public/Granted day:2015-04-02
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