Invention Application
WO2007002325A1 PYRROLO[2,3-B] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS
审中-公开
吡咯并[2,3-B]吡啶衍生物作为蛋白激酶抑制剂
- Patent Title: PYRROLO[2,3-B] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS
- Patent Title (中): 吡咯并[2,3-B]吡啶衍生物作为蛋白激酶抑制剂
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Application No.: PCT/US2006/024361Application Date: 2006-06-21
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Publication No.: WO2007002325A1Publication Date: 2007-01-04
- Inventor: IBRAHIM, Prahbha, N. , ARTIS, Dean, R. , BREMER, Ryan , MAMO, Shumeye , NESPI, Marika , ZHANG, Chao , ZHANG, Jiazhong , ZHU, Yong-Liang , TSAI, James , HIRTH, Klaus-Peter , BOLLAG, Gideon , SPEVAK, Wayne , CHO, Hanna , GILLETTE, Samuel, J. , WU, Guoxiam , ZHU, Hongyao , SHI, Shenghua
- Applicant: PLEXXIKON, INC. , IBRAHIM, Prahbha, N. , ARTIS, Dean, R. , BREMER, Ryan , MAMO, Shumeye , NESPI, Marika , ZHANG, Chao , ZHANG, Jiazhong , ZHU, Yong-Liang , TSAI, James , HIRTH, Klaus-Peter , BOLLAG, Gideon , SPEVAK, Wayne , CHO, Hanna , GILLETTE, Samuel, J. , WU, Guoxiam , ZHU, Hongyao , SHI, Shenghua
- Applicant Address: 91 Bolivar Drive, Suite A, Berkeley, CA 94710 US
- Assignee: PLEXXIKON, INC.,IBRAHIM, Prahbha, N.,ARTIS, Dean, R.,BREMER, Ryan,MAMO, Shumeye,NESPI, Marika,ZHANG, Chao,ZHANG, Jiazhong,ZHU, Yong-Liang,TSAI, James,HIRTH, Klaus-Peter,BOLLAG, Gideon,SPEVAK, Wayne,CHO, Hanna,GILLETTE, Samuel, J.,WU, Guoxiam,ZHU, Hongyao,SHI, Shenghua
- Current Assignee: PLEXXIKON, INC.,IBRAHIM, Prahbha, N.,ARTIS, Dean, R.,BREMER, Ryan,MAMO, Shumeye,NESPI, Marika,ZHANG, Chao,ZHANG, Jiazhong,ZHU, Yong-Liang,TSAI, James,HIRTH, Klaus-Peter,BOLLAG, Gideon,SPEVAK, Wayne,CHO, Hanna,GILLETTE, Samuel, J.,WU, Guoxiam,ZHU, Hongyao,SHI, Shenghua
- Current Assignee Address: 91 Bolivar Drive, Suite A, Berkeley, CA 94710 US
- Agency: WARBURG, Richard, J. et al.
- Priority: US60/692,960 20050622; US60/731,528 20051028
- Main IPC: C07D471/04
- IPC: C07D471/04 ; A61K31/435 ; C07C49/517 ; A61P35/00
Abstract:
Compounds of formula III which are active on protein kinases are described, as well as methods of using such compounds to treat diseases and conditions associated with aberrant activity of protein kinases.
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