Invention Application
- Patent Title: HETEROARYL COMPOUNDS AS BTK INHIBITORS AND USES THEREOF
- Patent Title (中): 作为BTK抑制剂的杂芳基化合物及其用途
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Application No.: PCT/US2014061455Application Date: 2014-10-21
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Publication No.: WO2015061247A2Publication Date: 2015-04-30
- Inventor: QIU HUI , CALDWELL RICHARD D , NEAGU CONSTANTIN , MOCHALKIN IGOR , LIU-BUJALSKI LESLEY , JONES REINALDO , TATE DEVON , JOHNSON THERESA L , GARDBERG ANNA
- Applicant: MERCK PATENT GMBH , QIU HUI , CALDWELL RICHARD D , NEAGU CONSTANTIN , MOCHALKIN IGOR , LIU-BUJALSKI LESLEY , JONES REINALDO , TATE DEVON , JOHNSON THERESA L , GARDBERG ANNA
- Assignee: MERCK PATENT GMBH,QIU HUI,CALDWELL RICHARD D,NEAGU CONSTANTIN,MOCHALKIN IGOR,LIU-BUJALSKI LESLEY,JONES REINALDO,TATE DEVON,JOHNSON THERESA L,GARDBERG ANNA
- Current Assignee: MERCK PATENT GMBH,QIU HUI,CALDWELL RICHARD D,NEAGU CONSTANTIN,MOCHALKIN IGOR,LIU-BUJALSKI LESLEY,JONES REINALDO,TATE DEVON,JOHNSON THERESA L,GARDBERG ANNA
- Priority: US201361893613 2013-10-21
- Main IPC: C07D213/81
- IPC: C07D213/81
Abstract:
The present invention relates to pyridine, pyrimidine, pyrazine, and pyridazine compounds, and pharmaceutically acceptable compositions thereof, useful as BTK inhibitors.
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