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1.发明公开QUINOLINE-CONTAINING $g(a)-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS 有权喹啉酮酰胺含基于抑制剂和半胱氨酸蛋白酶SERIN
公开(公告)号：EP1032393A1
公开(公告)日：2000-09-06
申请号：EP98952109.1
申请日：1998-10-07
发明人： CHATTERJEE, Sankar , MALLAMO, John, P. , DUNN, Derek, Douglas , JOSEF, Kurt, Allen , GU, Zi-Qiang , DAINES, Robert, A. , KINGSBURY, William, Dennis , PENDRAK, Israel , SHAM, Kelvin, C.
IPC分类号： A61K31/47 , A61K31/445 , C07D215/12 , C07D215/14 , C07D215/20 , C07D215/26
CPC分类号： C07D401/12 , C07D215/40 , C07D215/50 , C07D239/74 , C07D405/12 , C07D409/12 , C07D409/14 , C07D413/12 , C07D417/12
摘要： The present invention is directed to quinoline-containing α-ketoamide inhibitors of cysteine and serine proteases are disclosed. Methods for making these compounds, and methods for using the same are also disclosed.
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2.发明授权QUINOLINE-CONTAINING ALPHA-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS 有权喹啉含α-酮酰胺抑制剂基于半胱氨酸和SERIN蛋白酶
公开(公告)号：EP1032393B1
公开(公告)日：2006-08-09
申请号：EP98952109.1
申请日：1998-10-07
发明人： CHATTERJEE, Sankar , MALLAMO, John, P. , DUNN, Derek, Douglas , JOSEF, Kurt, Allen , GU, Zi-Qiang , DAINES, Robert, A. , KINGSBURY, William, Dennis , PENDRAK, Israel , SHAM, Kelvin, C.
IPC分类号： A61K31/47 , A61K31/445 , C07D417/12 , C07D413/12 , C07D409/14 , C07D405/12 , C07D401/12 , C07D215/50 , C07D409/12 , C07D239/74
CPC分类号： C07D401/12 , C07D215/40 , C07D215/50 , C07D239/74 , C07D405/12 , C07D409/12 , C07D409/14 , C07D413/12 , C07D417/12
摘要： The present invention is directed to quinoline-containing α-ketoamide inhibitors of cysteine and serine proteases are disclosed. Methods for making these compounds, and methods for using the same are also disclosed.
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公开(公告)号：EP1187607A1
公开(公告)日：2002-03-20
申请号：EP00941654.6
申请日：2000-06-22
IPC分类号： A61K31/40
CPC分类号： A61K31/404 , Y02A50/473
摘要： This invention relates to the use of compounds as inhibitors of the fatty acid synthase FabH useful in treating bacterial infections.
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