专利检索 ap:("Medivation Prostate Therapeutics LLC") AND inv:"GREENFIELD, Scott" 第 1 页

1.

发明公开
PROCESSES FOR THE SYNTHESIS OF DIARYLTHIOHYDANTOIN AND DIARYLHYDANTOIN COMPOUNDS 审中-公开

公开(公告)号：EP3329775A1

公开(公告)日：2018-06-06

申请号：EP18153287.0

申请日：2011-02-24

申请人： Medivation Prostate Therapeutics LLC

发明人： THOMPSON, Andrew , LAMBERSON, Carol , GREENFIELD, Scott , JAIN, Rajendra Parasmal , ANGELAUD, Remy

IPC分类号： A01N43/50 , A61K31/415 , C07D233/86 , C07D235/02 , C07C237/30

CPC分类号： C07D233/86 , C07C231/12 , C07C237/30 , C07D235/02

摘要： Processes are provided for the synthesis of diarylthiohydantoin and diarylhydantoin compounds, such as compounds of the formula:

wherein X, Y 1 , Y 2 , R 1 , and R 2 are as defined herein. Medicinal products containing the same find particular use in treating prostate cancer, including castration-resistant prostate cancer and/or hormone-sensitive prostate cancer.

2.

发明授权
PROCESSES FOR THE SYNTHESIS OF DIARYLTHIOHYDANTOIN AND DIARYLHYDANTOIN COMPOUNDS 有权
标题翻译：合成二芳基硫代嘌呤和二萘醌化合物的方法

公开(公告)号：EP2538785B1

公开(公告)日：2018-03-21

申请号：EP11748095.4

申请日：2011-02-24

申请人： Medivation Prostate Therapeutics LLC

发明人： THOMPSON, Andrew , LAMBERSON, Carol , GREENFIELD, Scott , JAIN, Rajendra, Parasmal , ANGELAUD, Remy

IPC分类号： A01N43/50 , A61K31/415 , C07D233/86 , C07D235/02

CPC分类号： C07D233/86 , C07C231/12 , C07C237/30 , C07D235/02

摘要： Processes are provided for the synthesis of diarylthiohydantoin and diarylhydantoin compounds. Medicinal products containing the same find particular use in treating prostate cancer, including castration-resistant prostate cancer and/or hormone-sensitive prostate cancer.