公开(公告)号：EP0934258B1

公开(公告)日：2001-08-29

申请号：EP97921762.7

申请日：1997-04-25

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： BAYER, Herbert ,  MÜLLER, Bernd ,  MÜLLER, Ruth ,  SAUTER, Hubert ,  GROTE, Thomas ,  GRAMMENOS, Wassilios ,  KIRSTGEN, Reinhard ,  OBERDORF, Klaus ,  PTOCK, Arne ,  GÖTZ, Norbert ,  RACK, Michael ,  RÖHL, Franz ,  AMMERMANN, Eberhard ,  HARRIES, Volker ,  LORENZ, Gisela ,  STRATHMANN, Siegfried

IPC: C07C271/28 ,  A01N47/24 ,  C07C327/58

CPC classification number: C07C327/58 ,  A01N47/24 ,  C07C271/28

Abstract: The invention pertains to phenylcarbamates of formula (I), wherein X is a direct bond, O or NR ; Z is O, S or NR ; R is hydrogen, alkyl or alkyl halide; R is substituted methyl or optionally substituted alkyl, alkenyl, alkinyl or cycloalkyl; R is optionally substituted alkyl, alkenyl or alkinyl; R is alkyl, alkenyl or alkinyl and, if X is NR , hydrogen also; R is hydrogen or optionally substituted alkyl, alkenyl, alkinyl, alkyl carbonyl or alkoxy carbonyl. The invention also pertains to methods for their preparation and agents containing them.

公开(公告)号：EP1085807A1

公开(公告)日：2001-03-28

申请号：EP99927805.4

申请日：1999-05-29

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MÜLLER, Bernd ,  SAUTER, Hubert ,  BAYER, Herbert ,  CULLMANN, Oliver ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GYPSER, Andreas ,  PTOCK, Arne ,  GÖTZ, Norbert ,  GROTE, Thomas ,  RACK, Michael ,  AMMERMANN, Eberhard ,  LORENZ, Gisela ,  STRATHMANN, Siegfried ,  SPEAKMAN, John-Bryan

IPC: A01N43/54

CPC classification number: C07D239/42 ,  A01N43/54

Abstract: The invention relates to the use of 2-(N-phenylamino)pyrimidines of formula (I) wherein the substituents have the following meanings: R1, R3 represent, independently of each other, cyano, C¿1?-C8-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, in which case the alkyl, alkenyl and alkinyl radicals can be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl; C3-C8-cycloalkyl or a group C(=NOR?x)Ry; and R2¿ represents halogen, C¿1?-C8-alkyl, C2-C6-alkenyl, C2-C6-alkinyl and the alkyl, alkenyl and alkinyl radicals can be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl; or R?1 and R2¿, together with the two carbon atoms with which they are bonded, form an anellated, partially unsaturated 4- to 8-membered ring which can be identically or differently substituted up to three times by C¿1?-C4-alkyl, halogen or C1-C4-alkoxycarbonyl, which can contain a carbonyl group and/or a double bond in addition to the multiple bond of the pyrimidine ring and/or which can be interrupted by O, S or N-(C1-C4-alkyl), the substituents R?4 to R8, Rx, Ry, Ra and Rb¿ having the meanings given in the description, as fungicides.

公开(公告)号：EP0858446B1

公开(公告)日：2001-03-07

申请号：EP96934776.4

申请日：1996-10-22

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MÜLLER, Bernd ,  SAUTER, Hubert ,  BAYER, Herbert ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  KIRSTGEN, Reinhard ,  OBERDORF, Klaus ,  RÖHL, Franz ,  GÖTZ, Norbert ,  RACK, Michael ,  MÜLLER, Ruth ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  HARRIES, Volker

IPC: C07C271/28 ,  C07C259/06 ,  C07C259/08 ,  C07C275/64 ,  A01N47/20 ,  A01N47/30 ,  A01N37/28

CPC classification number: C07C271/00 ,  C07C251/88 ,  C07C259/06 ,  C07C259/08 ,  C07C275/64

Abstract: The invention concerns phenylcarbamates of formula (I) in which the substituents and the index have the following meanings: R = cyano, nitro, trifluoromethyl, halogen, alkyl or alkoxy; m = 0, 1 or 2; R = alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkenyl and, if X stands for NR , additionally hydrogen; X is a direct bond, O or NR ; R = hydrogen, alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl; R = hydrogen, optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, cycloalkinyl, alkylcarbonyl or alkoxycarbonyl; R and R , independently of each other, stand for hydrogen, cyano, nitro, hydroxy, amino, halogen, optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkinyl, alkinyloxy, alkinylthio, alkinylamino, N-alkinyl-N-alkylamino, cycloalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocyclyl-N-alkylamino, aryl, aryloxy, arylthio, arylamino, N-aryl-N-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetarylamino or N-heteraryl-N-alkylamino; and R is one of the groups mentioned under R or a CR =NOR group. The invention further concerns processes and intermediate products for preparing these substances and their use as pesticides and fungicides.

公开(公告)号：EP0984944A1

公开(公告)日：2000-03-15

申请号：EP98924195.5

申请日：1998-05-05

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  MAYER, Guido ,  OTTEN, Martina ,  RACK, Michael ,  RHEINHEIMER, Joachim ,  WITSCHEL, Matthias ,  WESTPHALEN, Karl-Otto ,  MISSBLITZ, Ulf ,  WALTER, Helmut

IPC: C07D231/20 ,  A01N43/56

CPC classification number: C07D401/10 ,  A01N43/56 ,  C07D231/20 ,  C07D403/10 ,  C07D405/10 ,  C07D409/10 ,  C07D413/10 ,  C07D417/10

Abstract: The invention relates to 4-(3-alkenyl-benzoyl)-pyrazoles of formula (I), wherein the variables can have the following meanings: R1, R2 = hydrogen, nitro, halogen, cyano, rhodano, alkyl, halogen alkane, alkoxyalkyl, alkenyl, alkinyl, -OR?6, -OCOR7¿, -OSO¿2R?7, -SH, -S(O)nR8, -SO2OR6, -SO2NR?6R9, -NR9SO¿2R?7 or -NR9COR7; R3¿ = hydrogen, halogen, alkyl, halogen alkane, alkoxy, alkenyl, alkinyl; R4, R5 = hydrogen, nitro, halogen, cyano, rhodano, alkyl, halogen alkane, cycloalkyl, alkenyl, cycloalkenyl, alkinyl, alkythio, halogen alkoxy, -COR10, -CO2R?10, -COSR10, -CONR10R11, -C(R12)=NR13¿, -PO(OR?10) (OR11¿); optionally substituted alkyl, heterocyclyl, heterocyclylalkyl, phenyl, phenylalkyl, hetaryl or hetarylalkyl; or R?4 and R5¿ together form an alkandiyl chain which can be substituted and/or interrupted by a heteroatom; Q = a substituted position 4 bonded pyrazole. The invention further relates to the salts thereof, which can be used in agriculture. The invention also relates to a method for the production of compounds of formula (I), to agents containing said compounds and to the use of said derivatives or agents containing said compounds to control undesired plants.

公开(公告)号：EP0968188A1

公开(公告)日：2000-01-05

申请号：EP98913689.0

申请日：1998-03-09

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： SCHÄFER, Peter ,  HAMPRECHT, Gerhard ,  MENGES, Markus ,  MENKE, Olaf ,  RACK, Michael ,  ZAGAR, Cyrill ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf ,  WALTER, Helmut

IPC: C07D213/61 ,  A01N43/40

CPC classification number: C07D213/61 ,  A01N43/40

Abstract: Substituted 2-benz(o)ylpyridines of formula (I) and the salts thereof, wherein n = 0, 1; x = CO, CH2, CH(C1-C4-alkyl), CH-OH, CH-CN, CH-halogen, C(halogen)2, CH-CONH2, CH-CO-O(C1-C4-alkyl), CH-O(C1-C4-alkyl), C(CN) (C1-C4-alkyl); R1 = halogen, C¿1?-C4-halogen alkane, C1-C4-alkylthio, C1-C4-alkyl sulfinyl, C1-C4-alkyl sulfonyl; R?2¿ = H, halogen; R3 = H, NO¿2?, OH, halogen, C1-C4-alkoxy; R?4¿ = H, NO¿2?, OH, halogen, C1-C4-alkyl, C1-C4 halogen alkane, C1-C4-alkoxy; R?5¿ = H, NO¿2?, CN, halogen, C1-C8-alkyl, C3-C8-alkenyl,C3-C8-alkinyl, C3-C8-cycloalkyl, C1-C8-halogen alkane, C2-C8-halogen alkenyl, C2-C8-halogen alkane, C1-C4-alkoxy-C1-C4-alkyl, C2-C4-alkenyloxy-C1-C4-alkyl, C2-C4-alkinyloxy-C1-C4-alkyl, C1-C4-alkylthio-C1-C4-alkyl, C1-C4-alkylsulfinyl-C1-C4-alkyl, C1-C4-alkylsulfonyl-C1-C4-alkyl, cyano-C1-C8-alkyl, cyano-C2-C8-alkenyl, cyano-C3-C8-alkinyl, optionally substituted OH, SH, SO-H, -SO2-H, COOH or NH-COOH, -SO2Cl, -N(R?9, R10¿), -NH-SO¿2?-(C1-C8-alkyl), -N[-SO2-(C1-C8-alkyl)]2, -N(C1-C8-alkyl) [-SO2-(C1-C8-alkyl)], -SO2-N(R?9, R10¿), -O-CO-NH-R9, optionally substituted CHO, -O-CHO or -NH-CHO, NH-CO-NH-R9, -O-CS-NH¿2?, -OCS-N(C1-C8-alkyl)2, -CO-N(R?9, R10¿), -CS-N (R9, R10), -CO-NH-SO¿2?-(C1-C4-alkyl), -CO-N(C1-C4-alkyl), -SO2-(C1-C4-alkyl), hydroxycarbonyl-C1-C8-alkyl, (C1-C8-alkoxy)carbonyl-C1-C6-alkyl, -CH2-CH(halogen)-CO-N(R?9, R10¿), -CH¿2?-CH(halogen)-CN, -CH2-CH(halogen)-CO-(C1-C4-alkyl), optionally substituted -CH2-CH(halogen-COOH, -CH=C(halogen)-COOH or -CH=C(C1-C4-alkyl)-COOH, optionally substituted -CH=N-OH or -CH(-Y-R?15, -Z-R15¿), (II) or (III); R9, R10 = H, C¿1?-C8-alkyl, C3-C8-cycloalkyl, C2-C8-alkenyl, C3-C8-alkinyl, C1-C8-halogen alkane, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-alkylthio-C1-C4-alkyl, C1-C4-alkylsulfinyl-C1-C4-alkyl, C1-C4-alkylsulfonyl-C1-C4-alkyl, cyano-C1-C8-alkyl, hydroxycarbonyl-C1-C4-alkyl, (C1-C4-alkoxy)carbonyl-C1-C4-alkyl, (C3-C6-cycloalkoxy)carbonyl-C1-C4-alkyl, (C1-C4-alkoxy)carbonyl-C3-C7-cycloalkyl, C1-C4-alkoxy-(C1-C4)alkoxy)-carbonyl-C1-C4-alkyl, C1-C6-alkoxy, optionally substituted phenyl or phenyl-C1-C4-alkyl or R?9 + R10¿ together = optionally substituted tetramethylene, pentamethylene or ethylene oxyethylene chain; Y, Z = O, S; R15 = C1-C8-alkyl, C1-C8 halogen alkane, C1-C4-alkoxy-C1-C4-alkyl; R16-R21 = H, CN, C¿1?-C8-alkyl, C1-C4-alkoxy-C1-C4-alkyl, C1-C8-alkoxy, C1-C4-alkoxy-C1-C4-alkoxy, COOH, (C1-C8-alkoxy)carbonyl, CONH2, (C1-C8-alkyl)aminocarbonyl, di(C1-C8-alkyl)aminocarbonyl; R?6¿ = H, NO¿2?, halogen, optionally substituted OH or COOH; R?7¿ = H, NO¿2?, halogen, optionally substituted OH; excluding those compounds in (I) in wherein X = CH2 and R?5¿ = optionally substituted OH as well as R3, R7 = H or R1 = halogen as well as R?3, R4, R6, R7¿ = H. The invention further relates to the use of said substances as herbicides and for dessication/defoliation of plants.

公开(公告)号：EP0967867A1

公开(公告)日：2000-01-05

申请号：EP98905421.8

申请日：1998-02-12

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： BAYER, Herbert ,  SAUTER, Hubert ,  MÜLLER, Bernd ,  GRAMMENOS, Wassilios ,  KIRSTGEN, Reinhard ,  GYPSER, Andreas ,  PTOCK, Arne ,  GROTE, Thomas ,  RÖHL, Franz ,  RACK, Michael ,  GÖTZ, Roland ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  HARRIES, Volker

IPC: A01N33/24 ,  C07C259/02

CPC classification number: C07C259/02

Abstract: The invention relates to hydroximic acid halogenides of the formula (I) wherein the substituents have the following significance; X - NOCH3, CHOCH3 or CHCH3; Y - O or NH; R1 - halogen; R2 - optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or aryl; R3 - optionally substituted alkyl, alkoxyalkyl, cycloalkyl-alkyl, alkenyl and alkynyl and their salts. The invention also relates to a method for the production and use of said hydroximic acid halogenides.

公开(公告)号：EP0934258A1

公开(公告)日：1999-08-11

申请号：EP97921762.0

申请日：1997-04-25

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： BAYER, Herbert ,  MÜLLER, Bernd ,  MÜLLER, Ruth ,  SAUTER, Hubert ,  GROTE, Thomas ,  GRAMMENOS, Wassilios ,  KIRSTGEN, Reinhard ,  OBERDORF, Klaus ,  PTOCK, Arne ,  GÖTZ, Norbert ,  RACK, Michael ,  RÖHL, Franz ,  AMMERMANN, Eberhard ,  HARRIES, Volker ,  LORENZ, Gisela ,  STRATHMANN, Siegfried

IPC: C07C269 ,  A01N47 ,  C07C271 ,  C07C323 ,  C07C327

CPC classification number: C07C327/58 ,  A01N47/24 ,  C07C271/28

Abstract: The invention pertains to phenylcarbamates of formula (I), wherein X is a direct bond, O or NRa; Z is O, S or NRb; R1 is hydrogen, alkyl or alkyl halide; R2 is substituted methyl or optionally substituted alkyl, alkenyl, alkinyl or cycloalkyl; R3 is optionally substituted alkyl, alkenyl or alkinyl; R4 is alkyl, alkenyl or alkinyl and, if X is NRa, hydrogen also; R5 is hydrogen or optionally substituted alkyl, alkenyl, alkinyl, alkyl carbonyl or alkoxy carbonyl. The invention also pertains to methods for their preparation and agents containing them.

公开(公告)号：EP0920415A1

公开(公告)日：1999-06-09

申请号：EP97938899.0

申请日：1997-08-13

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： SCHÄFER, Peter ,  RACK, Michael ,  HAMPRECHT, Gerhard ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf ,  MENGES, Markus ,  ZAGAR, Cyrill ,  MENKE, Olaf

IPC: C07D213 ,  A01N43 ,  C07D405 ,  C07D409 ,  C07D411

CPC classification number: C07D405/10 ,  A01N43/40 ,  C07D213/71 ,  C07D405/12 ,  C07D409/10 ,  C07D411/10

Abstract: The present invention pertains to substituted 2-phenylpyridine I and the salts thereof of formula (I), where R1 = SH, SO¿2?NH2, C1-C2-alkylthio, C1-C6-alkyl-sulfinyl, C1-C6-akylsulfonyl, C1-C6alkylaminosulfonyl, Di-(C1-C6alkyl)aminosulfonyl; R?1, R3¿ = H, halogen; R4 = CN, OH, halogen, C¿1?-C6-alkoxy, possibly substituted OCH2-phenyl and R?5¿ have the meanings given in the description. The invention also relates to: the use of compounds (I) as herbicides or as plant dessicating/defoliating agents, the herbicides and the plant dessicating/defoliating agents containing compounds (I) as actives substances, the processes for controlling undesirable plant growth and for dessicating/defoliating plants using compounds (I), the processes for producing compounds (I), herbicides and plant dessicating/defoliating agents by compounds (I), as well as the intermerdiate products of formulae (IIa, V and VI).

公开(公告)号：EP0912524A1

公开(公告)日：1999-05-06

申请号：EP97923045.0

申请日：1997-05-09

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： RACK, Michael ,  RÖHL, Franz ,  AMMERMANN, Eberhard ,  HARRIES, Volker ,  LORENZ, Gisela ,  STRATHMANN, Siegfried ,  GROTE, Thomas ,  GRAMMENOS, Wassilios ,  KIRSTGEN, Reinhard ,  OBERDORF, Klaus ,  BAYER, Herbert ,  MÜLLER, Bernd ,  MÜLLER, Ruth ,  SAUTER, Hubert

IPC: C07D239 ,  A01N43

CPC classification number: C07D239/36 ,  A01N43/54 ,  C07D239/34

Abstract: 2-(O-[pyrimidin-4-yl] methylene oxy)phenyl acetic acid derivatives of general formula (I) and their salts and N oxides, in which R1 is halogen, alkyl or alkyl halide; R2 is hydrogen, amino, hydroxy, mercapto, halogen, possibly phenyl-substituted alkyl, alkyl halide, alkoxy alkyl, alkoxy, monoalkyl amino, dialkyl amino, alkylthio, alkyl sulphoxyl, alkylsulphonyl, cycloalkyl, trialkyl silyloxy or phenyl, phenoxy, phenoxy methyl, benzyloxy or heteroaryl possibly substituted in the aromatic ring, R2 being different from R1; R3 is hydrogen, cyano, halogen, C¿1?-C4 alkyl, C1-C4 alkyl halide or C1-C4 alkoxy, and Q is C(=CHCH3)-COOCH3 or C(=CHOCH3)-COOCH3, and their use in combatting noxious fungi and animal pests.

公开(公告)号：EP0888305A1

公开(公告)日：1999-01-07

申请号：EP97915376.0

申请日：1997-03-17

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： HARREUS, Albrecht ,  GÖTZ, Norbert ,  RACK, Michael ,  ISAK, Heinz ,  SCHÄFER, Peter

IPC: B01J23 ,  C07D213

CPC classification number: C07D213/61

Abstract: The invention concerns a process for preparing pyridyl-substituted N-phenylhydroxylamines of formula (II) by catalytically hydrogenating the corresponding nitro compounds in the presence of an N-substituted morpholine compound and rearranging the resultant hydroxylamine compounds to form pyridyl-4-fluoroaniline compounds of formula (I). The compounds of formula (I) are suitable as herbicides.