公开(公告)号：EP0973771A1

公开(公告)日：2000-01-26

申请号：EP98912471.4

申请日：1998-03-12

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MAYER, Guido ,  OTTEN, Martina ,  KARDORFF, Uwe ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  HILL, Regina, Luise ,  RHEINHEIMER, Joachim ,  WITSCHEL, Matthias ,  GÖTZ, Roland ,  RACK, Michael ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf ,  WALTER, Helmut

IPC: C07D417/04 ,  C07D417/14 ,  C07F9/6558 ,  A01N43/78 ,  A01N47/18 ,  A01N47/36

CPC classification number: C07D417/04 ,  A01N43/78 ,  A01N47/18 ,  A01N47/22 ,  A01N47/36 ,  A01N57/32 ,  C07D417/14 ,  C07F9/65586

Abstract: The invention relates to thiazolimines derivatives of formula (I), wherein the substituents have the following meanings: X, Y independently of each other stand for hydrogen, halogen, C1-C4-alkyl, C1-C4-haloalkyl, Z means hydrogen, C1-C8-alkyl, C2-C8-alkenyl, C2-C8-alkinyl, C1-C8-alkoxy, C1-C8-alkylthio, wherein these groups can be substituted by 1-5 halogen or C1-C4-alkoxy; aryl, hetaryl, benzyl, wherein these groups can be substituted with C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, halogen, nitro or cyano; or one of the following groups (a...); R1, R2 are hydrogen, halogen; C¿1?-C4-alkyl, C2-C4-alkenyl, C2-C4-alkinyl, wherein these groups can be substituted by 1-5 halogen or by C1-C4-alkoxy; n is 1 or 2; m is 0, 1 or 2, and R?3-R6¿ have the meaning cited in the application. The invention further relates to salts of compound I which can be used in agriculture.

公开(公告)号：EP0946514A1

公开(公告)日：1999-10-06

申请号：EP97953736.0

申请日：1997-12-04

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VOGELBACHER, Uwe, Josef ,  KEIL, Michael ,  KLINTZ, Ralf ,  WAHL, Joseph ,  WINGERT, Horst ,  KÖNIG, Hartmann ,  RACK, Michael ,  GÖTZ, Roland ,  TELES, Joaquim, Henrique

IPC: C07D231

CPC classification number: C07D231/22 ,  C07D231/20

Abstract: The invention relates to a method for producing n-substituted 3-hydroxypyrazoles of formula (I), wherein R1 stands for optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, aryl or heteroaryl and R?2 and R3¿ mean hydrogen, cyano, halogen and optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, aryl or heteroaryl, by oxidizing a corresponding pyrazolidin-3-ons.

公开(公告)号：EP0812317B1

公开(公告)日：1999-09-08

申请号：EP96916056.3

申请日：1996-05-13

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： GRAMMENOS, Wassilios ,  MÜLLER, Bernd ,  SAUTER, Hubert ,  OBERDORF, Klaus ,  KÖNIG, Hartmann ,  GÖTZ, Norbert ,  RACK, Michael ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried

IPC: C07D249/12 ,  C07D271/07 ,  C07D271/113 ,  C07D285/13 ,  C07D401/04 ,  C07D403/04 ,  C07D413/04 ,  C07D417/04 ,  A01N43/653 ,  A01N43/82

CPC classification number: C07D271/07 ,  A01N43/653 ,  A01N43/82 ,  C07D249/12 ,  C07D271/113 ,  C07D285/13 ,  C07D401/04

公开(公告)号：EP0934275A1

公开(公告)日：1999-08-11

申请号：EP97944808.0

申请日：1997-08-29

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： HAMPRECHT, Gerhard ,  GEBHARDT, Joachim ,  ISAK, Heinz ,  RACK, Michael ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter

IPC: C07D213

CPC classification number: C07D213/71

Abstract: Substituted thiopyridines having general formula (I), wherein n means 1 or 2, R1 means chlorine, C¿1?-C3 fluoralkyl, nitro or methylsulfonyl; a non-substituted or halogen, C1-C4 - alkoxy, C1-C4 aloxycarbonyl, di- (C1-C4-alkylamino) carbonyl, cyano or nitro substituted C1-C10-Alkyl, C2-C10-alkenyl or C2-C10 alkinyl radical, a C3-C8-cycloalkyl radical or a non-substituted in the phenyl part or hydrogen, C1-C3-alkyl, C1-C3-alkoxy, trifluormethyl, cyano or nitro substituted C1-C4-alkylene phenyl, phenyl or naphthyl radical.

Abstract translation: 其中n表示1或2，R1表示氯，C1-C3烷基，硝基或甲基磺酰基; 未取代或卤素，C 1 -C 4烷氧基，C 1 -C 4烷氧基，二（C 1 -C 4烷基氨基）羰基，氰基或硝基取代的C 1 -C 10烷基，C 2 -C 10链烯基或C 2 -C 10炔基 苯基部分中的未取代的C 3 -C 8环烷基或氢，C 1 -C 3烷基，C 1 -C 3烷氧基，三氟甲基，氰基或硝基取代的C 1 -C 4亚烷基苯基，苯基或萘基。

公开(公告)号：EP0882025A1

公开(公告)日：1998-12-09

申请号：EP97901621.0

申请日：1997-01-31

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： GRAMMENOS, Wassilios ,  BAYER, Herbert ,  GROTE, Thomas ,  KIRSTGEN, Reinhard ,  MÜLLER, Bernd ,  MÜLLER, Ruth ,  OBERDORF, Klaus ,  PTOCK, Arne ,  SAUTER, Hubert ,  RÖHL, Franz ,  RACK, Michael ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  HARRIES, Volker

IPC: C07D239 ,  A01N43

CPC classification number: C07D239/47 ,  A01N43/54 ,  C07D239/34

Abstract: The invention concerns pyrimidine derivatives of formula (I) in which the substituents have the following meanings: X is C(CO2CH3)=NOCH3, C(CONHCH3)=NOCH3, C(CO2CH3)=CHOCH3, C(CO2CH3)=CHCH3, N(CO2CH3)-OCH3; R?1 and R2¿, independently of each other, are hydrogen, C¿1?-C4 alkyl, C1-C4 alkyl halide or C1-C4 alkoxy; A is (i), the bond designated * being bonded to Y; R?3¿ is hydrogen, C¿1?-C4 alkyl, C1-C4 alkyl halide, phenoxy C1-C4 alkyl, C3-C6 cycloalkyl, cyano, C1-C4 alkoxy, hydroxy, halogen; R?4¿ is hydrogen, C¿1?-C8 alkyl, C1-C4 alkyl halide, C1-C6 cyanoalkyl, C1-C4 alkoxy-C1-C4 alkyl, C2-C4 alkenyloxy-C1-C4 alkyl, C1-C4 alkoxy halide-C1-C4 alkyl, C1-C4 oxoalkyl, C2-C4 alkenyl, C2-C4 alkinyl, C2-C4 alkenyl halide, C2-C4 alkinyl halide, C3-C6 cycloalkyl, C3-C6 cycloalkyl-C1-C4 alkyl, C1-C4 alkoxy; Y is hydrogen, hydroxy, halogen, optionally substituted aryl, hetaryl, cycloalkyl, cycloalkenyl, heterocyclyl, alkyl, alkenyl, alkinyl, alkyl halide, alkoxy, aryloxy, arylthio, hetaryloxy, hetarylthio, alkylthio or cycloalkyloxy; A not meaning -O- when X stands for C(CO2CH3)=CHOCH3. The invention also concerns the salts of these derivatives, a process and intermediate products for their preparation, and pesticides and fungicides containing them.

公开(公告)号：EP0851858A1

公开(公告)日：1998-07-08

申请号：EP96932485.0

申请日：1996-09-09

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： SCHÄFER, Peter ,  HAMPRECHT, Gerhard ,  HEISTRACHER, Elisabeth ,  MENKE, Olaf ,  ZAGAR, Cyrill ,  RACK, Michael ,  GÖTZ, Norbert ,  HARREUS, Albrecht ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut ,  MISSLITZ, Ulf

IPC: C07D213 ,  A01N43

CPC classification number: C07D213/61 ,  A01N43/40

Abstract: The invention concerns 2-phenylpyridines (I) and their salts, in which, n = 0, 1; R1 = halogen, C¿1?-C4 alkylhalide; R?2, R3¿ = H, halogen; R4 = CN, halogen; R5 = -CO-O-( C¿1?-C4 alkylene)-CO-OR?6¿, -CO-O-(C¿1?-C4 alkylene)-CO-N(R?7)R8¿, -O-(C¿1?-C4 alkylene)-CO-O-(C1-C4 alkylene)-CO-OR?6¿, -O-(C¿1?-C4 alkylene)-CO-O-(C1-C4 alkylene)-CO-N(R?7)R8¿, -S-(C¿1?-C4 alkylen)-CO-O-(C1-C4 alkylene)-CO-OR?6¿ or -S-(C¿1?-C4 alkylene)-CO-O-(C1-C4 alkylene)-CO-N(R?7)R8; R6¿ = H, C¿1?-C4 alkyl,(C1-C4 alkoxy)(C1-C4 alkyl), C2-C4 alkenyle, C3-C4 alkinyl; R?7¿ = H, C¿1?-C4 alkyl, carboxyl(C1-C4 alkyl), (C1-C4 alcoxycarbonyl)(C1-C4 alkyl); R?8¿ = H or C¿1?-C4 alkyl. Such compounds are suitable for use as herbicides and as plant desiccants/defoliants.

Abstract translation: 本发明涉及2-苯基吡啶（I）及其盐，其中n = 0,1; R1 =卤素，C1-C4烷基卤化物; R 2，R 3'= H，卤素; R4 = CN，卤素; R 5 = -CO-O-（C 1 -C 4亚烷基）-CO-OR 6，-CO-O-（C 1 -C 4亚烷基）-CO-N（R 7）R 8， （C 1 -C 4亚烷基）-CO-O-（C 1 -C 4亚烷基）-CO-OR 6'， - O-（C 1 -C 4亚烷基）-CO-O-（C1 （亚烷基）-CO-N（R 7）R 8，-S-（C 1 -C 4亚烷基）-CO-O-（C 1 -C 4亚烷基）-CO-OR 6或-S- （C 1 -C 4亚烷基）-CO-O-（C 1 -C 4亚烷基）-CO-N（R 7）R 8; （C 1 -C 4烷氧基）（C 1 -C 4烷基），C 2 -C 4烯烯基，C 3 -C 4炔基; R 6是H，C 1 -C 4烷基， （C 1 -C 4烷基），（C 1 -C 4烷氧基羰基）（C 1 -C 4烷基）; R 4为H，C 1 -C 4烷基。 R 8 = H或C 1 -C 4烷基。 这样的化合物适合用作除草剂和植物干燥剂/脱叶剂。

公开(公告)号：EP1863752A1

公开(公告)日：2007-12-12

申请号：EP06725104.1

申请日：2006-03-16

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： RACK, Michael ,  SMIDT, Sebastian, Peer ,  BUDICH, Manuel ,  MAYWALD, Volker ,  KEIL, Michael ,  WOLF, Bernd

IPC: C07C51/08 ,  C07C63/70 ,  C07C17/23 ,  C07C17/363 ,  C07C25/13

CPC classification number: C07C25/13 ,  C07C17/23 ,  C07C17/363 ,  C07C51/08 ,  C07C63/68

Abstract: The invention relates to a method for producing 5-halo-2,4,6-trifluoroisophthalic acid of formula (I), wherein X represents F, Cl, Br, or I, by hydrolysis of 5-halo-2,4,6-trifluoroisophthalodinitrile of formula (II). Said invention is characterised in that in a first step, isophthalodinitrile (II) or a solution containing isophthalodinitrile (II) is reacted with a concentrated sulphuric acid at room temperature in order to form a 5-haIo-2,4,6-trifluoroisophthalodiamide of general formula (III), and is, subsequently, heated and in a second step, isophthalic acid (I) is produced after additional heating and addition of water.

Abstract translation: 本发明涉及通过5-卤代-2,4,6,6-四氢吡啶的水解制备式（I）的5-卤代-2,4,6-三氟间苯二甲酸的方法，其中X代表F，Cl，Br或I （II）的三氟间苯二甲腈。 所述发明的特征在于，在第一步中，异佛尔酮二腈（II）或含有间苯二甲腈（II）的溶液在室温下与浓硫酸反应，以形成5-卤-2,4,6-三氟间苯二甲酰二胺 通式（III），随后加热，并且在第二步中，间苯二甲酸（I）在额外加热和加入水之后生成。

公开(公告)号：EP1863350A2

公开(公告)日：2007-12-12

申请号：EP06725266.8

申请日：2006-03-23

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEYN, Wolfgang ,  KAISER, Florian ,  POHLMAN, Matthias ,  BASTIAANS, Henricus Maria Martinus ,  BAUMANN, Ernst ,  RACK, Michael ,  ANSPAUGH, Douglas D. ,  COTTER, Henry Van Tuyl ,  CULBERTSON, Deborah L. ,  HOFMANN, Michael ,  HICKS, Carol

IPC: A01N41/06

CPC classification number: A01N41/06

Abstract: The present invention provides a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2- cyanobenzenesulfonamide compound of the general formula (I) where the variables R to R are as defined in claim 1.

Abstract translation: 本发明提供了一种保护种子免受土壤昆虫和所产生的植物的根和茎由土壤和叶面昆虫引起的方法，包括在播种之前和/或在萌芽之后使种子与通式（I）的2-氰基苯磺酰胺化合物接触， （I）其中变量R至R如权利要求1所定义。

公开(公告)号：EP1863349A1

公开(公告)日：2007-12-12

申请号：EP06725244.5

申请日：2006-03-22

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEYN, Wolfgang ,  KAISER, Florian ,  POHLMAN, Matthias ,  BASTIAANS, Henricus Maria Martinus ,  BAUMANN, Ernst ,  RACK, Michael ,  ANSPAUGH, Douglas D. ,  COTTER, Henry Van Tuyl ,  CULBERTSON, Deborah L. ,  HOFMANN, Michael ,  HICKS, Carol

IPC: A01N41/06

CPC classification number: A01N41/06 ,  A01N41/10

Abstract: The present invention provides a method for the protection of seeds from soil insects and of the seedlings’ roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/ or after pregermination with a sulphonyl compound of the general formula (I) where the variables R1 to R5 are as defined in claim 1.

公开(公告)号：EP1856122A2

公开(公告)日：2007-11-21

申请号：EP06724913.6

申请日：2006-03-02

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： GRAMMENOS, Wassilios ,  GROTE, Thomas ,  HÜNGER, Udo ,  LOHMANN, Jan Klaas ,  MÜLLER, Bernd ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHWÖGLER, Anja ,  RACK, Michael

IPC: C07D487/04 ,  A01N43/90

CPC classification number: C07D487/04

Abstract: The invention relates to 2-substituted 7-amino-azolopyrimidine of formula (I), wherein substituents have the following meanings: R1 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, Cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or akoxyalkinyl; R2 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, wherein a carbon chain in R1 and/or R2 are substitutable according to a description; R3 is halogen, Cyano, NRARB, hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phe- nylthio, benzyloxy, benzylthio, alkyl-S(O)m-; A N and CRx; Rx is hydrogen or one of above groups for R3. A method and intermediate products for producing said compounds, agents containing said compounds and the use thereof for combating plant-pathogen fungi are also disclosed.