专利检索 ap:("ABBOTT LABORATORIES") AND inv:"SCHMIDT, Robert, G." 第 1 页

1.

发明授权
2-AMINOOXAZOLE DERIVATIVES AS TRPVL ANTAGONISTS USEFUL FOR TREATING PAIN 有权
标题翻译： 2- AMINOOXAZOLDERIVATE AS疼痛SUITABLE的TRPV1拮抗剂的治疗

公开(公告)号：EP2220059B1

公开(公告)日：2011-08-03

申请号：EP08841479.2

申请日：2008-10-25

申请人： Abbott Laboratories

发明人： PERNER, Richard J. , KOENIG, John R. , DIDOMENICO, Stanley, Jr. , BAYBURT, Erol, K. , DAANEN, Jerome, F. , GOMTSYAN, Arthur, R. , KORT, Michael E. , KYM, Philip R. , VASUDEVAN, Anil , SCHMIDT, Robert, G. , VOIGHT, Eric

IPC分类号： C07D263/48 , C07D413/04 , C07D413/12 , A61K31/421 , A61P29/00

CPC分类号： C07D413/12 , C07D263/48 , C07D413/04

摘要： Compounds of formula (I) wherein R1, R2, R4, and W are defined in the description are TRPV1 antagonists with CNS penetration. Compositions comprising such compounds and methods for treating conditions and disorders using such compounds and compositions are also disclosed.

2.

发明公开
2-AMINOOXAZOLE DERIVATIVES AS TRPVL ANTAGONISTS USEFUL FOR TREATING PAIN 有权
标题翻译： 2-AMINOOXAZOLE DERIVATIVES TRPVL ANTAGONISTS用于治疗疼痛

公开(公告)号：EP2220059A1

公开(公告)日：2010-08-25

申请号：EP08841479.2

申请日：2008-10-25

申请人： Abbott Laboratories

发明人： PERNER, Richard J. , KOENIG, John R. , DIDOMENICO, Stanley, Jr. , BAYBURT, Erol, K. , DAANEN, Jerome, F. , GOMTSYAN, Arthur, R. , KORT, Michael E. , KYM, Philip R. , VASUDEVAN, Anil , SCHMIDT, Robert, G. , VOIGHT, Eric

IPC分类号： C07D263/48 , C07D413/04 , C07D413/12 , A61K31/421 , A61P29/00

CPC分类号： C07D413/12 , C07D263/48 , C07D413/04

摘要： Compounds of formula (I) wherein R1, R2, R4, and W are defined in the description are TRPV1 antagonists with CNS penetration. Compositions comprising such compounds and methods for treating conditions and disorders using such compounds and compositions are also disclosed.

摘要翻译： 其中R 1，R 2，R 4和W在说明书中定义的式（I）化合物是具有CNS穿透的TRPV1拮抗剂。还公开了包含此类化合物的组合物以及使用此类化合物和组合物治疗疾病和病症的方法。

3.

发明公开
NOVEL AZAHETEROCYCLIC AMIDES USEFUL FOR TREATING PAIN 审中-公开
标题翻译：疼痛治疗VBRAUCHBARE氮杂杂环酰胺

公开(公告)号：EP1646621A2

公开(公告)日：2006-04-19

申请号：EP04777733.9

申请日：2004-07-09

申请人： ABBOTT LABORATORIES

发明人： ZHENG, Guo Zhu , BROWN, Brian, S. , TURNER, Sean, C. , WHITE, Tammie, K. , SCHMIDT, Robert, G. , KOENIG, John, R. , LEE, Chih-Hung

IPC分类号： C07D401/04 , C07D401/12 , C07D487/08 , A61K31/4525 , A61K31/4995 , A61P25/04

CPC分类号： C07D401/04 , C07D487/08

摘要： The present invention relates to compounds of formula (I-VII) (I), or a pharmaceutically acceptable salt or prodrug thereof, in which A, L, R6, R7and R8 are defined herein. The present invention also relates to methods of trating pain using these compounds and pharmaceutical compositions including these compounds.