公开(公告)号：EP1150944A1

公开(公告)日：2001-11-07

申请号：EP00901791.4

申请日：2000-02-04

申请人： Aventis CropScience GmbH

发明人： CHARLES, Mark, David ,  FRANKE, Wilfried ,  GREEN, David, Eric,Aventis CropScience UK Limited ,  HOUGH, Thomas, Lawley,Aventis CropScience UK Ltd. ,  MITCHELL, Dale, Robert,Aventis CropScience UK Ltd ,  SIMPSON, Donald, James,Aventis CropScience UK Ltd ,  ATHERALL, John, F.,Aventis CropScience UK Ltd.

IPC分类号： C07C233/37 ,  C07D333/58 ,  C07D285/00 ,  C07D273/00 ,  C07C251/04 ,  A01N37/52 ,  A01N43/82

CPC分类号： C07D209/48 ,  A01N37/52 ,  A01N43/06 ,  A01N43/40 ,  A01N43/54 ,  A01N43/74 ,  A01N43/82 ,  A01N43/90 ,  A01N47/42 ,  C07C257/12 ,  C07C257/14 ,  C07D207/50 ,  C07D239/88 ,  C07D251/34 ,  C07D261/08 ,  C07D263/38 ,  C07D263/46 ,  C07D263/58 ,  C07D271/06 ,  C07D271/10 ,  C07D285/08 ,  C07D285/13 ,  C07D295/125 ,  C07D311/22 ,  C07D333/54 ,  C07D487/04 ,  C07D495/04 ,  C07F7/0812

摘要： The invention provides fungicidal compounds of formula (I) and salts thereof wherein: R1 is alkyl, alkenyl, alkynyl, carbocyclyl or heterocyclyl, each of which may be substituted, or hydrogen; R?2 and R3¿, which may be the same or different, are any group defined for R1; cyano; acyl; -OR?a or -SRa¿, where Ra is alkyl, alkenyl, alkynyl, carbocyclyl or heterocyclyl, each of which may be substituted; or R?2 and R3, or R2 and R1¿, together with their interconnecting atoms may form a ring, which may be substituted; R4 is alkyl, alkenyl, alkynyl, carbocyclyl or heterocyclyl, each of which may be substituted; hydroxy; mercapto; azido; nitro; halogen; cyano; acyl; optionally substituted amino; cyanato; thiocyanato; -SF¿5?; -OR?a; -SRa¿ or -Si(Ra)3; m is 0 to 3; when present R5, which may be the same or different to any other R5, is any group defined for R4; R6 is optionally substituted carbo- or heterocylclyl; and A is a defined linking group, or -A-R?6 and R5¿ together with benzene ring M form an optionally substituted fused ring system.

摘要翻译： 本发明提供了式（I）的杀真菌化合物及其盐，其中：R 1为各自可被取代的烷基，烯基，炔基，碳环基或杂环基或氢; R 2和R 3可以相同或不同，是对R1定义的任何基团; 氰基; 酰基; 其中Ra是烷基，烯基，炔基，碳环基或杂环基，它们中的每一个可以被取代; 或R 2和R 3或R 2和R 1'与它们的相互连接的原子一起可形成可被取代的环; R4是烷基，链烯基，炔基，碳环基或杂环基，它们中的每一个可以被取代; 羟基; 巯基; 叠氮; 硝基; 卤素; 氰基; 酰基; 任选取代的氨基; 氰酸酯; 氰硫基; -SF¿5?; -OR一个？; -SRa或-Si（Ra）3; m是0至3; 当存在时，与任何其它R5可以相同或不同的R5是R4中定义的任何基团; R6是任选取代的碳 - 或杂环基; A是定义的连接基团，或者-A-R 6和R 5'与苯环M一起形成任选取代的稠合环体系。