公开(公告)号：EP0986549A1

公开(公告)日：2000-03-22

申请号：EP98930724.4

申请日：1998-05-25

申请人： Bayer Aktiengesellschaft

发明人： DYKER, Hubert ,  SCHERKENBECK, Jürgen ,  HARDER, Achim ,  MENCKE, Norbert ,  VON SAMSON-HIMMELSTJERNA, Georg

IPC分类号： C07D273/00 ,  C07D413/14 ,  C07D413/10 ,  A61K31/395

CPC分类号： C07D273/00 ,  C07D413/10 ,  C07D413/14

摘要： The invention relates to novel desoxycyclodepsipeptides of formula (I) in which C=X?1, C=X2, C=X3¿ and C=X4 independently of each other respectively represent one of the CO, CS or CH¿2? groups, with at least one of these groups representing CH2. The invention also relates to their mixtures and derivatives. Said compounds are produced from cyclodepsipeptides having 24 ring members formed by alternating α-amino carboxylic acids and α-hydroxy carboxylic acids by complete or partial chemoselective reduction of the carbonyl groups of the amide function into methylene groups, using suitable reduction methods. The desoxycyclodepsipeptides produced according to the invention have an anthelmintic effect.

公开(公告)号：EP0973387A1

公开(公告)日：2000-01-26

申请号：EP98913576.9

申请日：1998-02-23

申请人： Bayer Aktiengesellschaft

发明人： JUSTUS, Karl ,  LENZ, Jürgen, Georg ,  NENTWIG, Günther ,  SCHERKENBECK, Jürgen ,  DAMBACH, Martin ,  WENDLER, Gernot

IPC分类号： A01N37/06 ,  A01N37/10 ,  A01N37/08 ,  A01N37/04 ,  A01N25/00

CPC分类号： A01N37/08 ,  A01N25/006 ,  A01N37/04 ,  A01N37/10 ,  A01N47/36 ,  A01N37/02 ,  A01N2300/00

摘要： The use is disclosed of a new combination of carboxylic acids as attractant for controlling cockroaches, as well as corresponding agents and devices containing this combination.

公开(公告)号：EP1090031A1

公开(公告)日：2001-04-11

申请号：EP99927953.2

申请日：1999-06-11

申请人： Bayer Aktiengesellschaft

发明人： SCHERKENBECK, Jürgen ,  DYKER, Hubert ,  PLANT, Andrew ,  HARDER, Achim ,  VON SAMSON HIMMELSTJERNA, Georg

IPC分类号： C07K11/02 ,  C07D273/00 ,  A61K38/15

CPC分类号： C07K11/02 ,  A61K38/00

摘要： The invention relates to new substituted cyclooctadepsipeptides of formula (I) wherein R1, R2, m and n are as defined in the description, a method for their preparation and their use for fighting endoparasites, as well as drugs containing them as active ingredients.

摘要翻译： 本发明涉及式（I）的新的取代的环十八缩酚酸肽，其中R 1，R 2，m和n如说明书中所定义，其制备方法及其用于抵抗体内寄生虫的用途，以及含有它们作为活性成分的药物。