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1.发明公开
公开(公告)号：EP1301188A2
公开(公告)日：2003-04-16
申请号：EP01957894.7
申请日：2001-06-26
发明人： HARDER, Achim , VON SAMSON-HIMMELSTJERNA, Georg , KRÜGER, Bernd-Wieland , MEHLHORN, Heinz , SCHMIDT, Jürgen
IPC分类号： A61K31/5375 , A01N43/84 , A01N47/38
CPC分类号： A61K31/5375
摘要： The invention relates to agents that contain certain active substances according to formula (I), wherein R?1 to R10¿ are defined as in the claims, that are useful as repellents. The invention further relates to the use of said agents for preventing humans or animals from being infected with the infective stages of parasitic flatworms (platyhelminths).
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2.发明公开
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3.发明公开
公开(公告)号：EP1317562A2
公开(公告)日：2003-06-11
申请号：EP01974211.3
申请日：2001-08-24
发明人： VON SAMSON-HIMMELSTJERNA, Georg , HARDER, Achim , WUNDERLICH, Frank , SCHMITT-WREDE, Hans-Peter , SAEGER, Beate
IPC分类号： C12Q1/25 , C12Q1/02 , C12Q1/68 , C12N15/00 , C07K14/435
CPC分类号： G01N33/502 , C07K14/4354 , C07K14/705 , C07K14/723 , C12Q1/6888 , G01N33/5008 , G01N33/5014 , G01N33/5085 , G01N33/5308 , G01N33/6872 , G01N2333/4353 , G01N2333/4719 , G01N2333/705
摘要： The invention relates to test systems that are based on transmembrane receptors from helminths and arthropods and to their use for identifying and characterizing substances that are effective against helminths, arthropods or that have an effect on the calcium metabolism of organisms and/or cells. The invention further relates to the use of a specific ligand in said test system and to the use thereof as an anthelminthic or arthropodan active substance.
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公开(公告)号：EP1208199A2
公开(公告)日：2002-05-29
申请号：EP00956159.8
申请日：2000-06-30
IPC分类号： C12N15/12
CPC分类号： C07K14/4354 , A61K38/00
摘要： The invention relates to DNA which codes for β-tubulin from nematodes of the Strongylidae family, to the polypeptide coded by this DNA, to the use of the DNA for diagnosing anthelmintic resistance in the nematodes concerned and for identifying parasitic nematode species, to the use of the β-tubulin as a component of a vaccine and to a method for identifying novel anthelmintic or antibiotic compounds.
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公开(公告)号：EP1169328A2
公开(公告)日：2002-01-09
申请号：EP00925111.7
申请日：2000-03-13
发明人： HALLENBACH, Werner , HARDER, Achim , TURBERG, Andreas , HANSEN, Olaf , VON SAMSON-HIMMELSTJERNA, Georg
IPC分类号： C07H19/00
CPC分类号： C07H17/08
摘要： The invention relates to novel avermectin derivatives of formula (I), in which R?1, R2, R3 and R4¿ have the meanings defined in the description. The invention also relates to various methods for producing them, to agents containing them and to their use for producing agents for combating ecto- and endoparasites in animals.
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6.发明公开DESOXYCYCLODEPSIPEPTIDE UND IHRE VERWENDUNG ZUR BEKÄMPFUNG VON ENDOPARASITEN 失效DESOXYCYCLODEPSIPEPTIDE和使用控制体内寄生虫
公开(公告)号：EP0986549A1
公开(公告)日：2000-03-22
申请号：EP98930724.4
申请日：1998-05-25
发明人： DYKER, Hubert , SCHERKENBECK, Jürgen , HARDER, Achim , MENCKE, Norbert , VON SAMSON-HIMMELSTJERNA, Georg
IPC分类号： C07D273/00 , C07D413/14 , C07D413/10 , A61K31/395
CPC分类号： C07D273/00 , C07D413/10 , C07D413/14
摘要： The invention relates to novel desoxycyclodepsipeptides of formula (I) in which C=X?1, C=X2, C=X3¿ and C=X4 independently of each other respectively represent one of the CO, CS or CH¿2? groups, with at least one of these groups representing CH2. The invention also relates to their mixtures and derivatives. Said compounds are produced from cyclodepsipeptides having 24 ring members formed by alternating α-amino carboxylic acids and α-hydroxy carboxylic acids by complete or partial chemoselective reduction of the carbonyl groups of the amide function into methylene groups, using suitable reduction methods. The desoxycyclodepsipeptides produced according to the invention have an anthelmintic effect.
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7.发明授权6-SUBSTITUIERTE 1,2,4A,5A,8A,8B-HEXAHYDRO- UND 1,2,3,4,4A,5A,8A,8B-OKTAHYDRO-6H-PYRROLO[3',4':4,5]FURO[3,2-B]PYRID-8(7H)-ON DERIVATE UND IHRE VERWENDUNG ZUR BEKÄMPFUNG VON ENDOPARASITEN 失效6-取代的1,2,4a，5A，8A，8B六氢AND -1,2,3，5A，8A，8B八氢-6H-吡咯并[3”，4' ：4,5] 呋喃并[3,2-B]吡啶-8（7H） - 酮衍生物及其用途FOR CONTROLLING体内寄生虫
公开(公告)号：EP0986564B1
公开(公告)日：2003-10-15
申请号：EP98929269.3
申请日：1998-04-29
IPC分类号： C07D491/14 , A61K31/44
CPC分类号： C07D491/14
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8.发明公开ENDOPARASITIZIDE SYNERGISTISCHE KOMBINATION ENTHALTEND CYCLISCHEN DEPSIPEPTIDEN UND PIPERAZINEN 有权Endoparasiticides协同组合含环酯肽和哌嗪
公开(公告)号：EP1189615A2
公开(公告)日：2002-03-27
申请号：EP00940235.5
申请日：2000-05-04
IPC分类号： A61K31/495 , A61K38/15
CPC分类号： A61K31/495 , A61K38/15 , A61K2300/00
摘要： The invention relates to the use of piperazines for potentiating the endoparasiticidal action of cyclic depsipeptides in endoparasiticidal agents. Said depsipeptides are comprised of amino acids and hydroxycarboxylic acids serving as ring structural elements and having 24 ring atoms. The invention also relates to agents of this type and to the use of piperazines and cyclic depsipeptides, said depsipeptides being comprised of amino acids and hydroxycarboxylic acids serving as ring structural elements and having 24 ring atoms, in order to produce endoparasiticidal agents.
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9.发明公开
公开(公告)号：EP1318795A2
公开(公告)日：2003-06-18
申请号：EP01969321.7
申请日：2001-06-26
发明人： HARDER, Achim , VON SAMSON-HIMMELSTJERNA, Georg , KRÜGER, Bernd-Wieland , MEHLHORN, Heinz , SCHMIDT, Jürgen
IPC分类号： A61K31/00
CPC分类号： A61K31/221 , A61K31/223
摘要： The invention relates to agents containing specific active ingredients that act as repellents and to their use for preventing humans or animals from being infected with parasitic flatworms (platyhelminths).
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10.发明公开ANTHELMINTIKA ZUR VERHINDERUNG VON PARASITÄREN INFEKTIONEN BEI MENSCH UND TIER II 审中-公开驱虫为了预防感染人畜寄生虫II
公开(公告)号：EP1309320A2
公开(公告)日：2003-05-14
申请号：EP01945311.7
申请日：2001-06-25
发明人： HARDER, Achim , VON SAMSON-HIMMELSTJERNA, Georg , KRÜGER, Bernd-Wieland , MEHLHORN, Heinz , SCHMIDT, Jürgen
IPC分类号： A61K31/16 , A61K31/4453 , A61P33/00
CPC分类号： A61K31/4453 , A61K31/16
摘要： The invention relates to agents containing particular active ingredients which can be used as repellents, and the use thereof to prevent humans or animals being infected by the stages of infection of parasitic flatworms (platyhelminths). Said active ingredients are cyclic or acyclic amides.
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