公开(公告)号：EP2473476A1

公开(公告)日：2012-07-11

申请号：EP10745569.3

申请日：2010-08-18

申请人： Bayer CropScience AG

发明人： MORADI, Wahed Ahmed ,  LUI, Norbert ,  DOCKNER, Michael ,  JAGUSCH, Thomas

IPC分类号： C07C201/12 ,  C07C209/68 ,  C07C205/06 ,  C07C205/12 ,  C07C231/12 ,  C07F5/02 ,  C07C233/15

CPC分类号： C07F5/027 ,  C07C231/12 ,  C07C233/15

摘要： The present invention relates to a process for producing substituted biphenyls by reacting aryl halides with tetraarylborates in the presence of palladium catalysts.

公开(公告)号：EP2245001A1

公开(公告)日：2010-11-03

申请号：EP08866428.9

申请日：2008-12-16

申请人： Bayer CropScience AG

发明人： LUI, Norbert ,  WOLLNER, Thomas ,  WIESCHEMEYER, Jürgen ,  DOCKNER, Michael ,  HEINRICH, Jens-Dietmar

IPC分类号： C07C227/16 ,  C07C229/30

CPC分类号： C07C227/16 ,  C07C253/30 ,  C07C229/30 ,  C07C255/30

摘要： The present invention relates to a method for the production of 2-fluoroacyl-3-amino-acrylic acid derivatives by reacting fluorinated carboxylic acids with dialkylaminoacrylic acid derivatives and acid halogenides.

公开(公告)号：EP2245001B1

公开(公告)日：2013-03-20

申请号：EP08866428.9

申请日：2008-12-16

申请人： Bayer CropScience AG

发明人： LUI, Norbert ,  WOLLNER, Thomas ,  WIESCHEMEYER, Jürgen ,  DOCKNER, Michael ,  HEINRICH, Jens-Dietmar

IPC分类号： C07C227/16 ,  C07C229/30

CPC分类号： C07C227/16 ,  C07C253/30 ,  C07C229/30 ,  C07C255/30

公开(公告)号：EP2257530B1

公开(公告)日：2011-10-12

申请号：EP09713907.5

申请日：2009-02-12

申请人： Bayer CropScience AG

发明人： DOCKNER, Michael ,  RIECK, Heiko

IPC分类号： C07D213/82 ,  C07D231/14

CPC分类号： C07D213/82 ,  C07D231/14

摘要： The present invention relates to a process for preparing substituted biphenylanilides of the formula (I) which comprises reacting a compound of formula (II) in the presence of a base and of a palladium catalyst selected from the group of: a) palladium-triarylphosphine or -trialkylphosphine complex with palladium in the zero oxidation state, b) salt of palladium in the presence of triarylphospine or trialkylphosphine as a complex ligand or c) metallic palladium, optionally applied to support, in the presence of triarylphosphine or trialkylphosphine, in a solvent, with a diphenylborinic acid according to formula (III).

公开(公告)号：EP2280932A1

公开(公告)日：2011-02-09

申请号：EP09741817.2

申请日：2009-04-24

申请人： Bayer CropScience AG

发明人： DOCKNER, Michael ,  RIECK, Heiko ,  MORADI, Wahed Ahmed ,  LUI, Norbert

IPC分类号： C07C231/12

CPC分类号： C07C231/12 ,  C07C233/15

摘要： The present invention relates to a process for preparing substituted biphenylanilides of the formula (I), wherein R
1 is a protected amino group which comprises reacting a compound of formula (II), in the presence of a base and of a palladium catalyst in a solvent, with an organoboron compound of formula (III).

摘要翻译： 本发明涉及一种制备式I取代的联苯酰苯胺的方法，其中R 1是被保护的氨基，其包括使式II化合物在碱和钯催化剂存在下在溶剂中与有机硼化合物 的式（III）