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1.发明公开
公开(公告)号：EP2167495A1
公开(公告)日：2010-03-31
申请号：EP08759100.4
申请日：2008-06-07
发明人： RÖHRIG, Susanne , HÄRTER, Michael , GNOTH, Mark, Jean , VON DEGENFELD, Georges , DITTRICH-WENGENROTH, Elke , BUCHMÜLLER, Anja , ALLERHEILIGEN, Swen , PERZBORN, Elisabeth , GERDES, Christoph , SCHLEMMER, Karl-Heinz , AKBABA, Metin
IPC分类号： C07D409/12 , A61K31/4412 , A61P7/02
CPC分类号： C07D409/12 , C07D413/14
摘要： The invention relates to novel substituted oxazolidinones of the formula (I), a method for the production thereof, the use thereof for the treatment and/or prophylaxis of diseases, and the use thereof for the production of medications for the treatment and/or prophylaxis of diseases, particularly of thromboembolic disorders. Formula (I) where R' = formula (Ia), (Ib), (Ic), (Id), (Ie), (If), (Ig), (Ih) or (Ii).
摘要翻译： 本发明涉及式（I）的新型取代的恶唑烷酮类，其制备方法，其用于治疗和/或预防疾病的用途，以及其用于制备用于治疗和/或预防的药物的用途 的疾病，特别是血栓栓塞性疾病。 其中R'=式（Ia），（Ib），（Ic），（Id），（Ie），（If），（Ig），（Ih）或（Ii）的式（I）
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2.发明授权NEUE, ZYKLISCH SUBSTITUIERTE FUROPYRIMIDIN-DERIVATE UND IHRE VERWENDUNG ZUR BEHANDLUNG VON KARDIOVASKULÄREN ERKRANKUNGEN 有权新的环状结构的取代furopyrimidine衍生物及其用于治疗心血管疾病治疗
公开(公告)号：EP1966218B1
公开(公告)日：2010-07-14
申请号：EP06840964.8
申请日：2006-12-08
发明人： LAMPE, Thomas , BECKER, Eva-Maria , KAST, Raimund , BECK, Hartmut , JESKE, Mario , SCHUHMACHER, Joachim , STOLL, Friederike , KLEIN, Martina , AKBABA, Metin , KNORR, Andreas , STASCH, Johannes-Peter , BÄRFACKER, Lars , HILLISCH, Alexander , KARIG, Gunter , MEININGHAUS, Mark , SCHLEMMER, Karl-Heinz , SCHOHE-LOOP, Rudolf
IPC分类号： C07D491/04 , A61K31/519 , A61P9/00
CPC分类号： C07D491/04
摘要： The invention relates to novel, cyclic substituted furopyrimidine derivatives represented by formula (I), to methods for the production thereof, to the use thereof for treating and/or for the prophylaxis of illnesses and to the use thereof for producing medicaments for treating and/or for the prophylaxis of diseases, in particular for treating and/or for the prophylaxis of cardiovascular diseases.
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3.发明公开AMINOACYL-PRODRUGS ALS ARZNEIMITTELWIRKSTOFF FÜR THROMBOEMBOLISCHE ERKRANKUNGEN 审中-公开AMINOACYL-PRODRUGS ALS ARZNEIMITTELWIRKSTOFFFÜRTHROMBOEMBOLISCHE ERKRANKUNGEN
公开(公告)号：EP2167500A1
公开(公告)日：2010-03-31
申请号：EP08773746.6
申请日：2008-06-28
发明人： LERCHEN, Hans-Georg , KRENZ, Ursula , HÄRTER, Michael , GNOTH, Mark, Jean , VON DEGENFELD, Georges , DITTRICH-WENGENROTH, Elke , BUCHMÜLLER, Anja , RÖHRIG, Susanne , ALLERHEILIGEN, Swen , PERZBORN, Elisabeth , GERDES, Christoph , SCHLEMMER, Karl-Heinz , AKBABA, Metin
IPC分类号： C07D413/14 , A61K31/422 , A61P7/02
CPC分类号： C07D413/14
摘要： The present invention relates to prodrug derivatives of 5-chloro-N-({(5S)-3-[2-fluoro-4-(3- oxomopholin-4-yl)phenyl]-2-oxo-l,3-oxazolidin-5-yl}methyl)thiophene-2-carboxamide, to processes for preparation thereof, to the use thereof for treatment and/or prophylaxis of disorders, and to the use thereof for production of medicaments for treatment and/or prophylaxis of disorders, especially of thromboembolic disorders.
摘要翻译： 本发明涉及5-氯-N - （{（5S）-3- [2-氟-4-（3-氧代吗啉-4-基）苯基] -2-氧代-1,3-恶唑烷的前药衍生物 -5-基}甲基）噻吩-2-甲酰胺，涉及其制备方法，其用于治疗和/或预防疾病的用途，及其用于制备用于治疗和/或预防疾病的药物的用途， 特别是血栓栓塞性疾病。
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公开(公告)号：EP1945634B1
公开(公告)日：2011-01-19
申请号：EP06806430.2
申请日：2006-10-20
发明人： RÖHRIG, Susanne , POHLMANN, Jens , ARNDT, Sabine , JESKE, Mario , AKBABA, Metin , PERZBORN, Elisabeth , GERDES, Christoph , SCHLEMMER, Karl-Heinz
IPC分类号： C07D413/14 , A61K31/422 , A61P7/02
CPC分类号： C07D413/14
摘要： The present invention relates to novel 1,4-phenylenebisoxazolidine derivatives, to processes for their preparation, to their use for the treatment and/or prophylaxis of diseases and to their use for the production of medicaments for the treatment and/or prophylaxis of diseases, especially of thromboembolic disorders.
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5.发明公开SUBSTITUIERTE DIHYDROPYRAZOLONE ALS HEMMER DER HIF-PROLYL-4-HYDROXYLASE 有权代入为HIF脯氨酰4-羟化酶抑制剂dihydropyrazolones
公开(公告)号：EP2265602A1
公开(公告)日：2010-12-29
申请号：EP09733899.0
申请日：2009-04-11
发明人： JESKE, Mario , FLAMME, Ingo , STOLL, Friederike , BECK, Hartmut , AKBABA, Metin
IPC分类号： C07D401/14 , C07D403/14 , C07D413/14 , A61K31/506 , A61K31/5355 , A61K31/553 , A61P9/00 , A61P13/12 , A61P7/06
CPC分类号： C07D403/14 , C07D401/14 , C07D413/14
摘要： The present application relates to novel substituted dihydropyrazolone derivatives, to methods for the preparation thereof, to the use thereof for the treatment and/or prophylaxis of diseases and to the use thereof for the production of medicines for the treatment and/or prophylaxis of diseases, in particular cardiovascular and hematological diseases, kidney diseases, and for the promotion of wound healing.
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