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公开(公告)号:EP2188275A2
公开(公告)日:2010-05-26
申请号:EP08803004.4
申请日:2008-08-12
发明人: SCHNAUBELT, Jürgen , FACHINGER, Thomas , KONRAD, Michael , KRUEGER, Thomas , MERTEN, Joern , REICHEL, Carsten , RENNER, Svenja , SCHMID, Rolf , STEHLE, Emanuel , WERNER, Bianca
IPC分类号: C07D401/14 , C07D211/58 , C07D309/12 , C07C69/96
CPC分类号: C07D401/14 , C07C69/96 , C07C2601/14 , C07D211/58 , C07D309/12
摘要: The present invention relates to a process for preparing compounds of the general formula (I) in which R1 and R2 are defined as mentioned in the description, the pharmaceutically acceptable salts thereof and the solvates thereof, which can be prepared starting from compounds of the general formula (II) in which R1 is defined as mentioned in the description.
摘要翻译: 制备式(I)化合物的方法,其中R 1和R 2如说明书中所定义。
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公开(公告)号:EP2268622A1
公开(公告)日:2011-01-05
申请号:EP09723550.1
申请日:2009-03-19
发明人: DURAN, Adil , GOEPPER, Stefan , HALMER, Joerg , KONRAD, Michael
IPC分类号: C07D239/42
CPC分类号: C07D239/42
摘要: The present invention relates to a method of making pyrimidines of formula (III), wherein X1, X2, R1 and R2 have the meanings as defined herein.
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公开(公告)号:EP2195294A1
公开(公告)日:2010-06-16
申请号:EP08803003.6
申请日:2008-08-12
发明人: PACHUR, Kathrin , GOEPPER, Stefan , HUCHLER, Günther , KONRAD, Michael , MAIER, Kathrin , RALL, Werner , RIES, Uwe Jörg , ZOPF, Andreas
IPC分类号: C07D211/58 , C07D401/04 , C07D401/14 , C07C229/42
CPC分类号: C07D211/58 , C07C229/42 , C07D401/04 , C07D401/14
摘要: The present invention relates to a process for preparing compounds of the general formula (I) in which R1.1, R11.2, R1.3 and R2 are defined as mentioned in the description, the pharmaceutically acceptable salts thereof and the solvates thereof, which can be prepared starting from compounds of the general formula (II) in which R1.1, R1.2 and R1.3 are defined as mentioned in the description.
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