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1.发明授权SUBSTITUTED BENZAMIDES WITH ACTIVITY TOWARDS EP4 RECEPTORS 有权SUBSTITUIERTE BENZAMIDE MITAKTIVITÄTGEGENÜBEREP4-REZEPTOREN
公开(公告)号：EP2953927B1
公开(公告)日：2016-11-16
申请号：EP14706498.4
申请日：2014-02-07
IPC分类号： C07C255/57 , C07D213/81 , C07D239/26 , C07C235/56 , A61K31/192 , A61K31/277 , A61K31/4418 , A61K31/4453 , A61P19/02 , A61P19/08 , A61P29/00 , C07C233/81 , C07C235/42
CPC分类号： C07D213/81 , C07C233/81 , C07C235/42 , C07C235/56 , C07C255/57 , C07C2601/04 , C07C2601/14 , C07D239/26
摘要： The present invention belongs to the field of EP4 receptor ligands. More specifically it refers to compounds of general formula (I) having great affinity and selectivity for the EP4 receptor. The invention also refers to the process for their preparation, to their use as medicament for the treatment and/or prophylaxis of diseases or disorders mediated by the EP4 receptor as well as to pharmaceutical compositions comprising them.
摘要翻译： 本发明属于EP4受体配体领域。 更具体地，其是指对EP4受体具有很大亲和性和选择性的通式（I）的化合物。 本发明还涉及其制备方法，用作药物用于治疗和/或预防由EP4受体介导的疾病或病症以及包含它们的药物组合物。
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公开(公告)号：EP2953927A1
公开(公告)日：2015-12-16
申请号：EP14706498.4
申请日：2014-02-07
IPC分类号： C07C255/57 , C07D213/81 , C07D239/26 , C07C235/56 , A61K31/192 , A61K31/277 , A61K31/4418 , A61K31/4453 , A61P19/02 , A61P19/08 , A61P29/00
CPC分类号： C07D213/81 , C07C233/81 , C07C235/42 , C07C235/56 , C07C255/57 , C07C2601/04 , C07C2601/14 , C07D239/26
摘要： The present invention belongs to the field of EP4 receptor ligands. More specifically it refers to compounds of general formula (I) having great affinity and selectivity for the EP4 receptor. The invention also refers to the process for their preparation, to their use as medicament for the treatment and/or prophylaxis of diseases or disorders mediated by the EP4 receptor as well as to pharmaceutical compositions comprising them.
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