N-Benzoyl urea compounds, antitumorous compositions containing them, and process for their preparation
    2.
    发明公开
    N-Benzoyl urea compounds, antitumorous compositions containing them, and process for their preparation 失效
    含有它们的制备抗肿瘤这些组合物和方法的N-苯甲酰脲化合物。

    公开(公告)号:EP0226104A2

    公开(公告)日:1987-06-24

    申请号:EP86116595.9

    申请日:1986-11-28

    摘要: An N-benzoyl urea compound having the formula:
    wherein X is a hydrogen atom, a halogen atom or a nitro group, n is an integer of from 1 to 3, and Q is
    wherein Y, is an unsubstituted or substituted alkyl group, or an alkoxy or alkoxycarbonyl group with its alkyl moiety unsubstituted or substituted, Y 2 is a hydrogen atom, a halogen atom, a nitro group, an unsubstituted or substituted alkyl group, or an alkoxy or alkoxycarbonyl group with its alkyl moiety unsubstituted or substituted, Z is a hydrogen atom, a halogen atom, a trifluoromethyl group or a nitro group, and each of A and B is =CH- or a nitrogen atom, provided that one of A and B is =CH- and the other is a nitrogen atom, with the provisos (1) that when Q is
    where when X is a hydrogen atom and Y, is an alkyl group, Z is not a hydrogen atom, a halogen atom nor a trifluoromethyl group, and (2) that when Q is
    wherein A is a nitrogen atom and Y, is a trifluoromethyl group, Y 2 is other than a hydrogen atom.

    An O-(N-alkoxy-pyridinecarboximidoyl)phosphate, a process for producing the same, and an insecticidal or acaricidal composition containing the same
    3.
    发明公开
    An O-(N-alkoxy-pyridinecarboximidoyl)phosphate, a process for producing the same, and an insecticidal or acaricidal composition containing the same 失效
    O-(N-烷氧基 - pyridincarboximidoyl)磷酸酯,其制备方法和杀虫或含有它的杀螨组合物的方法。

    公开(公告)号:EP0065039A1

    公开(公告)日:1982-11-24

    申请号:EP81302009.6

    申请日:1981-05-07

    摘要: An O-(N-alkoxy-pyridinecarboximidoyl)-phosphate is represented by the following formula:
    wherein X is a halogen atom, a lower alkyl group, a lower acyloxy group. a trifluoromethyl group or a nitro group; Y is an oxygen atom or a sulfur atom; R is a lower alkyl group; n is an integer of 0 to 3; and Z 1 and Z 2 are each a lower alkoxy group, a lower alkylthio group, a phenyl group which may be substituted by a lower alkyl group, a phenoxy group, a haloalkoxy group or a lower alkylamino group.
    The compound of formula (I) is useful as an active ingredient of insecticides or acaricides and is produced by reacting an N-alkoxy-pyridinecarboximidic acid having the formula (A):
    wherein X, R and n are as defined above with a phosphoric halide having the formula (B):
    wherein Hal is a halogen atom and Y, Z, and Z. are as defined above in the presence of an alkaline material.

    摘要翻译: O-(N-alkoxypyridinecarboximidoyl)磷酸酯由下式表示: worin X是卤原子,低级烷基,低级酰氧基,三氟甲基或硝基; Y是氧原子或硫原子; R是低级烷基; n为0〜3的整数; Z1和Z2各自为一个低级烷氧基,低级烷硫基,可被低级烷基,苯氧基,卤代烷氧基或低级烷基氨基取代的苯基。 式(I)的化合物可用作在杀虫剂或杀螨剂的活性成分,并通过使成N-烷氧基 - pyridinecarboximidic酸具有下式(A)制备: worin X,R和n如以上所定义 具有式(B)磷酸卤化物: worin Hal为卤原子,Y,Z 1和Z 2如上述在碱性物质的存在下定义。