公开(公告)号：EP1391450A4

公开(公告)日：2005-08-17

申请号：EP01930006

申请日：2001-05-09

申请人： KUREHA CHEMICAL IND CO LTD

发明人： ITO ATSUSHI ,  SUDO KEIICHI ,  WATANABE TSUMORU ,  KUSANO NOBUYUKI ,  ARAKI NOBUYUKI ,  EIZUKA TAKAYOSHI ,  NIIZEKI YOSHITAKA

IPC分类号： A01N43/40 ,  C07D207/32 ,  C07D207/325 ,  C07D207/335 ,  C07D213/38 ,  C07D213/61 ,  C07D231/12 ,  C07D233/54 ,  C07D233/64 ,  C07D239/26 ,  C07D241/12 ,  C07D241/16 ,  C07D249/08 ,  C07D277/32 ,  C07D401/12 ,  C07D405/12 ,  C07D413/12

CPC分类号： C07D207/325 ,  A01N43/40 ,  C07D207/335 ,  C07D213/38 ,  C07D213/61 ,  C07D231/12 ,  C07D233/64 ,  C07D239/26 ,  C07D241/12 ,  C07D241/16 ,  C07D249/08 ,  C07D277/32 ,  C07D401/12 ,  C07D405/12 ,  C07D413/12

摘要： An N-(heterocycle-methyl)alkylamine derivative which is one represented by the following general formula (I) or an acid addition salt thereof. [In the formula, R1 represents a heterocycle containing at least one nitrogen atom as a heteroatom and optionally having one or more substituents on the ring; R2 represents hydrogen, etc.; R3 represents C¿1-5? alkyl, etc. and R?4¿ represents C¿1-5? alkyl, etc., provided that when R?4¿ is C¿1-5? alkyl or C1-5 halogenoalkyl, then a carbon atom of R?3¿ may be bonded to a carbon atom of R4 to form a ring structure; m is an integer of 1 to 3; and R5 represents, e.g., cycloalkyl represented by the following formula (III) (wherein Y and Z each represents hydrogen, etc.; p is an integer of 2 to 5; and the groups represented by CYZ may be the same or different) provided that when m is 1 and R4 is hydrogen, then R5 is cycloalkyl represented by the formula (III).]