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公开(公告)号：EP2462122A1
公开(公告)日：2012-06-13
申请号：EP10743082.9
申请日：2010-08-05
发明人： CHALTIN, Patrick , DEBYSER, Zeger , DE MAEYER, Marc , MARCHAND, Arnaud , MARCHAND, Damien , SMETS, Wim , VOET, Arnout , CHRIST, Frauke
IPC分类号： C07D239/26 , C07D239/42 , A61K31/505 , A61P31/18
CPC分类号： C07D491/052 , C07D239/26 , C07D239/38 , C07D239/42 , C07D401/04 , C07D401/14 , C07D403/04 , C07D405/04 , C07D409/04 , C07D413/14 , C07D417/04
摘要： The present invention relates to a series of novel compounds having antiviral activity, more specifically HIV (Human Immunodeficiency Virus) replication inhibiting properties. The invention also relates to methods for the preparation of such compounds, as well as to novel intermediates useful in one or more steps of such syntheses. The invention also relates to pharmaceutical compositions comprising an effective amount of such compounds as active ingredients. This invention further relates to the use of such compounds as medicines or in the manufacture of a medicament useful for the treatment of animals suffering from viral infections, in particular HIV infection. This invention further relates to methods for the treatment of viral infections in animals by the administration of a therapeutical amount of such compounds, optionally combined with one or more other drugs having antiviral activity.
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公开(公告)号：EP4363438A1
公开(公告)日：2024-05-08
申请号：EP22801342.1
申请日：2022-07-04
CPC分类号： C07K14/001 , G16B15/20 , C07K19/00
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公开(公告)号：EP2640705A2
公开(公告)日：2013-09-25
申请号：EP11781819.5
申请日：2011-11-15
发明人： CHALTIN, Patrick , CHRIST, Frauke , DEBYSER, Zeger , DE MAEYER, Marc , MARCHAND, Arnaud , MARCHAND, Damien , VOET, Arnout
IPC分类号： C07D221/06 , C07D221/08 , C07D221/10 , C07D401/04 , C07D417/04 , C07D471/04 , C07D471/14 , C07D487/04 , C07D491/048 , C07D491/06 , C07D495/04 , C07D495/14 , C07D519/00 , A61P31/00 , A61K31/435 , A61K31/4355 , A61K31/437 , A61K31/519
CPC分类号： A61K31/519 , A61K31/437 , A61K31/473 , A61K45/06 , C07D221/06 , C07D221/08 , C07D221/10 , C07D221/16 , C07D401/04 , C07D417/04 , C07D471/04 , C07D471/14 , C07D487/04 , C07D487/14 , C07D491/048 , C07D491/06 , C07D491/16 , C07D495/04 , C07D495/14 , C07D519/00 , A61K2300/00
摘要： The present invention relates to compounds of formula (A), as further defined herein, having antiviral activity, more specifically HIV (Human Immunodeficiency Virus) replication inhibiting 5 properties. The invention also relates to pharmaceutical compositions comprising an effective amount of such compounds as active ingredients. The invention further relates to the use of such compounds, optionally combined with one or more other drugs having antiviral activity, for the treatment of animals suffering from viral infections, in particular HIV infection.
摘要翻译： 本发明涉及如本文进一步定义的式（A）化合物，其具有抗病毒活性，更具体地说是HIV（人类免疫缺陷病毒）复制抑制性质。 本发明还涉及包含有效量的这种化合物作为活性成分的药物组合物。 本发明进一步涉及这种化合物的用途，其任选地与一种或多种具有抗病毒活性的其它药物组合用于治疗患有病毒感染，特别是HIV感染的动物。
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公开(公告)号：EP2516008A1
公开(公告)日：2012-10-31
申请号：EP10801407.7
申请日：2010-12-20
发明人： CARLENS, Gunter , CHALTIN, Patrick , CHRIST, Frauke , DEBYSER, Zeger , MARCHAND, Arnaud , MARCHAND, Damien , VOET, Arnout , DE MAEYER, Marc
IPC分类号： A61P31/18 , A61K31/519 , C07D487/04
CPC分类号： C07D487/04
摘要： The present invention relates to compounds of formula (A) as defined herein having antiviral activity, more specifically HIV (Human Immunodeficiency Virus) replication inhibiting properties. The invention also relates to pharmaceutical 5 compositions comprising an effective amount of such compounds as active ingredients. This invention further relates to the use of such compounds as medicines or in the manufacture of a medicament useful for the treatment of animals suffering from viral infections, in particular HIV infection. This invention further relates to methods for the treatment of viral infections in animals by the 10 administration of a therapeutical amount of such compounds, optionally combined with one or more other drugs having antiviral activity.
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5.发明授权
公开(公告)号：EP2430029B1
公开(公告)日：2018-01-10
申请号：EP10721773.9
申请日：2010-05-17
发明人： BARDIOT, Dorothée , CHALTIN, Patrick , CHRIST, Frauke , DEBYSER, Zeger , DE MAEYER, Marc , MARCHAND, Arnaud , MARCHAND, Damien , VOET, Arnout
IPC分类号： C07D495/04 , A61K31/4365 , A61P31/18
CPC分类号： C07D495/20 , A61K31/4365 , A61K31/4375 , A61K45/06 , C07D495/04 , C07D495/14
摘要： The present invention relates to a series of compounds having antiviral activity, more specifically HIV (Human Immunodeficiency Virus) replication inhibiting properties. The invention also relates to methods for the preparation of such compounds, as well as to novel intermediates useful in one or more steps of such syntheses. The invention also relates to pharmaceutical compositions comprising an effective amount of such compounds as active ingredients. This invention further relates to the use of such compounds as medicines or in the manufacture of a medicament useful for the treatment of animals suffering from viral infections, in particular HIV infection. This invention further relates to methods for the treatment of viral infections in animals by the administration of a therapeutic amount of such compounds, optionally combined with one or more other drugs having anti-viral activity.
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公开(公告)号：EP2516008B1
公开(公告)日：2014-04-16
申请号：EP10801407.7
申请日：2010-12-20
发明人： CARLENS, Gunter , CHALTIN, Patrick , CHRIST, Frauke , DEBYSER, Zeger , MARCHAND, Arnaud , MARCHAND, Damien , VOET, Arnout , DE MAEYER, Marc
IPC分类号： A61P31/18 , A61K31/519 , C07D487/04
CPC分类号： C07D487/04
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7.发明公开
公开(公告)号：EP2430029A1
公开(公告)日：2012-03-21
申请号：EP10721773.9
申请日：2010-05-17
发明人： BARDIOT, Dorothée , CHALTIN, Patrick , CHRIST, Frauke , DEBYSER, Zeger , DE MAEYER, Marc , MARCHAND, Arnaud , MARCHAND, Damien , VOET, Arnout
IPC分类号： C07D495/04 , A61K31/4365 , A61P31/18
CPC分类号： C07D495/20 , A61K31/4365 , A61K31/4375 , A61K45/06 , C07D495/04 , C07D495/14
摘要： The present invention relates to a series of compounds of formula (A) having antiviral activity, more specifically HIV (Human Immunodeficiency Virus) replication inhibiting properties. The invention also relates to methods for the preparation of such compounds, as well as to novel intermediates useful in one or more steps of such syntheses. The invention also relates to pharmaceutical compositions comprising an effective amount of such compounds as active ingredients. This invention further relates to the use of such compounds as medicines or in the manufacture of a medicament useful for the treatment of animals suffering from viral infections, in particular HIV infection. This invention further relates to methods for the treatment of viral infections in animals by the administration of a therapeutical amount of such compounds, optionally combined with one or more other drugs having anti-viral activity.
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