公开(公告)号：EP0034945A3

公开(公告)日：1982-04-21

申请号：EP81300767

申请日：1981-02-24

申请人： MAY & BAKER LIMITED

发明人： Hatton, Leslie Roy ,  Parnell, Edgar William ,  Roberts, David Alan

IPC分类号： C07D231/38 ,  A01N43/56 ,  C07C109/00 ,  C07C87/52 ,  C07C87/60 ,  C07C121/78 ,  C07C79/12 ,  C07C121/52

CPC分类号： C07D231/38 ,  A01N43/56 ,  A01N47/02 ,  C07C243/00 ,  C07C255/00

摘要： N-Phenylpyrazole derivatives of the formula:-
(wherein each of R 5 and R 6 represents a C 1 -C 4 alkyl or alkoxy radical, a trifluoromethyl, trifluoromethoxy, nitro, cyano or primary amino radical, or a fluorine, chlorine or bromine atom, each of R', R' and R 9 represents a hydrogen atom, a C 1 -C 4 alkyl or alkoxy radical, a trifluoromethyl, trifluoromethoxy, nitro, cyano or primary amino radical or a fluorine, chlorine or bromine atom, or R 5 , R 7 , R' and R 9 each represents a hydrogen atom and R 6 represents a trifluoromethoxy or trifluoromethyl radical, and R 10 represents a cyano radical or substituted carbamoyl radical -CONHR", wherein R" represents a methyl or ethyl radical) have been found to possess useful herbicidal properties. All such N-phenylpyrazole derivatives with the exception of 5-amino-4-cyano-1-(2,4-dichlorophenyl)pyrazole and 5-amino-4-cyano-1- (4-chloro-2-methylphenyl)pyrazole are new compounds. Herbicidal compositions containing such N-phenylpyrazole derivatives are described and also processes for the prepararation of the new compounds.

公开(公告)号：EP0034945A2

公开(公告)日：1981-09-02

申请号：EP81300767.1

申请日：1981-02-24

申请人： MAY & BAKER LIMITED

发明人： Hatton, Leslie Roy ,  Parnell, Edgar William ,  Roberts, David Alan

IPC分类号： C07D231/38 ,  A01N43/56

CPC分类号： C07D231/38 ,  A01N43/56 ,  A01N47/02 ,  C07C243/00 ,  C07C255/00

摘要： N-Phenylpyrazole derivatives of the formula:-
(wherein each of R 5 and R 6 represents a C 1 -C 4 alkyl or alkoxy radical, a trifluoromethyl, trifluoromethoxy, nitro, cyano or primary amino radical, or a fluorine, chlorine or bromine atom, each of R', R' and R 9 represents a hydrogen atom, a C 1 -C 4 alkyl or alkoxy radical, a trifluoromethyl, trifluoromethoxy, nitro, cyano or primary amino radical or a fluorine, chlorine or bromine atom, or R 5 , R 7 , R' and R 9 each represents a hydrogen atom and R 6 represents a trifluoromethoxy or trifluoromethyl radical, and R 10 represents a cyano radical or substituted carbamoyl radical -CONHR", wherein R" represents a methyl or ethyl radical) have been found to possess useful herbicidal properties. All such N-phenylpyrazole derivatives with the exception of 5-amino-4-cyano-1-(2,4-dichlorophenyl)pyrazole and 5-amino-4-cyano-1- (4-chloro-2-methylphenyl)pyrazole are new compounds. Herbicidal compositions containing such N-phenylpyrazole derivatives are described and also processes for the prepararation of the new compounds.

摘要翻译： 下式的N-苯基吡唑衍生物： - （其中R 5和R 6各自表示C 1 -C 4烷基或烷氧基，三氟甲基，三氟甲氧基，硝基，氰基或伯氨基，或 氟，氯或溴原子，R 7，R 8和R 9各自表示氢原子，C 1 -C 4烷基或烷氧基，三氟甲基，三氟甲氧基，硝基，氰基或伯氨基，或 氟，氯或溴原子，或R 5，R 7，R 8和R 9各自表示氢原子，R 6表示三氟甲氧基或三氟甲基，R 1， 已经发现，<0>表示氰基或取代的氨基甲酰基-CONHR 1（其中R 1表示甲基或乙基）具有有用的除草性质。 所有这样的N-苯基吡唑衍生物除了5-氨基-4-氰基-1-（2,4-二氯苯基）吡唑和5-氨基-4-氰基-1-（4-氯-2-甲基苯基）吡唑是 新化合物。 描述了含有这种N-苯基吡唑衍生物的除草组合物，以及制备新化合物的方法。

公开(公告)号：EP0034945B1

公开(公告)日：1985-08-07

申请号：EP81300767.1

申请日：1981-02-24

申请人： MAY & BAKER LIMITED

发明人： Hatton, Leslie Roy ,  Parnell, Edgar William ,  Roberts, David Alan

IPC分类号： C07D231/38 ,  A01N43/56

CPC分类号： C07D231/38 ,  A01N43/56 ,  A01N47/02 ,  C07C243/00 ,  C07C255/00

公开(公告)号：EP0278742A3

公开(公告)日：1989-11-15

申请号：EP88301103.3

申请日：1988-02-10

申请人： MAY & BAKER LIMITED

发明人： Geach, Neil Jonathan ,  Gilmour, James ,  Hatton, Leslie Roy ,  Smith, Philip Henry Gaunt

IPC分类号： C07D211/86 ,  C07D309/32 ,  C07D221/20 ,  C07C49/792 ,  C07C79/36 ,  A01N43/40 ,  A01N43/16 ,  A01N35/00

CPC分类号： C07D309/32 ,  A01N35/06 ,  A01N37/42 ,  A01N41/10 ,  A01N43/16 ,  A01N43/18 ,  A01N43/28 ,  A01N43/30 ,  A01N43/40 ,  A01N43/42 ,  A01N43/86 ,  A01N47/22 ,  C07C45/54 ,  C07C49/792 ,  C07C49/813 ,  C07C49/83 ,  C07C49/835 ,  C07C49/84 ,  C07C205/55 ,  C07C323/56 ,  C07C2601/14 ,  C07D211/86

摘要： A 2-benzoylcyclic-1,3-dione derivative of the formula:
wherein X represents methylene, oxygen, sulphur or -NR⁴-, Y represents -C(R⁵) (R⁶)- or oxygen, R¹ represents hydrogen or alkyl optionally substituted by halogen or represents cycloalkyl, R² represents hydrogen or R⁷ or R¹ and R² together represent alkylene, R³ represents halogen, hydroxy, carboxy, nitro, cyano or amino or carbamoyl (which may be substituted by one or two alkyl groups) , alkoxycarbonyl, alkanoyl, or alkanoylamino, R, RO, RS, RSO or RSO₂ in which R represents alkyl optionally substituted by halogen, R⁴ represents hydrogen or alkyl or alkoxycarbonyl, R⁵ represents hydrogen or alkyl or alkoxycarbonyl, R⁶ represents hydrogen or alkyl, R⁷ represents alkyl which may be substituted by halogen or alkylthio or by a group (R⁸) n -phenyl-S-, or represents cycloalkyl or tetrahydrothiapyran-3-yl or represents a group (R⁸) n -phenyl- ­in which R⁸ represents a halogen, hydroxy, carboxy, nitro or cyano, or amino or carbamoyl (which may be substituted by one or two alkyl groups), alkoxycarbonyl or alkanoyl or alkanoylamino or R, RO, RS, RSO or RSO₂ in which R represents alkyl which is optionally substituted by halogen, m is zero or 1 to 5 and n is zero or 1 to 5, provided that when X represents methylene, and Y represents -C(R⁵) (R⁶)- ­then R¹ and R² do not simultaneously represent hydrogen or alkyl and salts thereof are useful as herbicides.

摘要翻译： 下式的2-苯甲酰基-1,3-二酮衍生物：其中X代表亚甲基，氧，硫或-NR 4 - ，Y代表-C（R 5）（R 6） - 或氧，R 1表示氢或任选被卤素取代的烷基或代表环烷基，R 2表示氢或R 7或R 1和R 2一起表示亚烷基，R 3表示 卤素，羟基，羧基，硝基，氰基或氨基或氨基甲酰基（其可以被一个或两个烷基取代），烷氧基羰基，烷酰基或烷酰基氨基，R，RO，RS，RSO或RSO 2，其中R表示任选被 卤素，R 4表示氢或烷基或烷氧基羰基，R 5表示氢或烷基或烷氧基羰基，R 6表示氢或烷基，R 7表示可以被卤素或烷硫基取代的烷基或由 基团（R 8）n-苯基-S-，或代表环烷基或四氢噻喃-3-基或代表（R 8）n-苯基 - ，其中R 8表示卤素，羟基，羧基 ，硝基或c 氨基或氨基甲酰基（其可以被一个或两个烷基取代），烷氧基羰基或烷酰基或烷酰基氨基或R，RO，RS，RSO或RSO 2，其中R表示任选被卤素取代的烷基，m为零或 1至5，n为0或1至5，条件是当X表示亚甲基，Y表示-C（R 5）（R 6））时，则R 1和R 2不同时 代表氢或烷基，其盐可用作除草剂。

公开(公告)号：EP0278742A2

公开(公告)日：1988-08-17

申请号：EP88301103.3

申请日：1988-02-10

申请人： MAY & BAKER LIMITED

发明人： Geach, Neil Jonathan ,  Gilmour, James ,  Hatton, Leslie Roy ,  Smith, Philip Henry Gaunt

IPC分类号： C07D211/86 ,  C07D309/32 ,  C07D221/20 ,  C07C49/792 ,  C07C79/36 ,  A01N43/40 ,  A01N43/16 ,  A01N35/00

CPC分类号： C07D309/32 ,  A01N35/06 ,  A01N37/42 ,  A01N41/10 ,  A01N43/16 ,  A01N43/18 ,  A01N43/28 ,  A01N43/30 ,  A01N43/40 ,  A01N43/42 ,  A01N43/86 ,  A01N47/22 ,  C07C45/54 ,  C07C49/792 ,  C07C49/813 ,  C07C49/83 ,  C07C49/835 ,  C07C49/84 ,  C07C205/55 ,  C07C323/56 ,  C07C2601/14 ,  C07D211/86

摘要： A 2-benzoylcyclic-1,3-dione derivative of the formula:
wherein X represents methylene, oxygen, sulphur or -NR⁴-, Y represents -C(R⁵) (R⁶)- or oxygen, R¹ represents hydrogen or alkyl optionally substituted by halogen or represents cycloalkyl, R² represents hydrogen or R⁷ or R¹ and R² together represent alkylene, R³ represents halogen, hydroxy, carboxy, nitro, cyano or amino or carbamoyl (which may be substituted by one or two alkyl groups) , alkoxycarbonyl, alkanoyl, or alkanoylamino, R, RO, RS, RSO or RSO₂ in which R represents alkyl optionally substituted by halogen, R⁴ represents hydrogen or alkyl or alkoxycarbonyl, R⁵ represents hydrogen or alkyl or alkoxycarbonyl, R⁶ represents hydrogen or alkyl, R⁷ represents alkyl which may be substituted by halogen or alkylthio or by a group (R⁸) n -phenyl-S-, or represents cycloalkyl or tetrahydrothiapyran-3-yl or represents a group (R⁸) n -phenyl- ­in which R⁸ represents a halogen, hydroxy, carboxy, nitro or cyano, or amino or carbamoyl (which may be substituted by one or two alkyl groups), alkoxycarbonyl or alkanoyl or alkanoylamino or R, RO, RS, RSO or RSO₂ in which R represents alkyl which is optionally substituted by halogen, m is zero or 1 to 5 and n is zero or 1 to 5, provided that when X represents methylene, and Y represents -C(R⁵) (R⁶)- ­then R¹ and R² do not simultaneously represent hydrogen or alkyl and salts thereof are useful as herbicides.

摘要翻译： 下式的2-苯甲酰基-1,3-二酮衍生物：其中X代表亚甲基，氧，硫或-NR 4 - ，Y代表-C（R 5）（R 6） - 或氧，R 1表示氢或任选被卤素取代的烷基或代表环烷基，R 2表示氢或R 7或R 1和R 2一起表示亚烷基，R 3表示 卤素，羟基，羧基，硝基，氰基或氨基或氨基甲酰基（其可以被一个或两个烷基取代），烷氧基羰基，烷酰基或烷酰基氨基，R，RO，RS，RSO或RSO 2，其中R表示任选被 卤素，R 4表示氢或烷基或烷氧基羰基，R 5表示氢或烷基或烷氧基羰基，R 6表示氢或烷基，R 7表示可以被卤素或烷硫基取代的烷基或由 基团（R 8）n-苯基-S-，或代表环烷基或四氢噻喃-3-基或代表（R 8）n-苯基 - ，其中R 8表示卤素，羟基，羧基 ，硝基或c 氨基或氨基甲酰基（其可以被一个或两个烷基取代），烷氧基羰基或烷酰基或烷酰基氨基或R，RO，RS，RSO或RSO 2，其中R表示任选被卤素取代的烷基，m为零或 1至5，n为0或1至5，条件是当X表示亚甲基，Y表示-C（R 5）（R 6））时，则R 1和R 2不同时 代表氢或烷基，其盐可用作除草剂。

公开(公告)号：EP0269238A1

公开(公告)日：1988-06-01

申请号：EP87309141.7

申请日：1987-10-15

申请人： MAY & BAKER LIMITED

发明人： Feldwick, Graham Alan ,  Hatton, Leslie Roy ,  Hewett, Richard Henry ,  Pedgrift, Brian Leslie

IPC分类号： A01N43/50 ,  C07D233/92 ,  C07D233/90

CPC分类号： C07D233/90 ,  A01N43/50

摘要： The invention provides a method of regulating the growth of a plant using a compound of the formula:
wherein R¹ represents alkyl or phenyl optionally substituted by halogen, alkyl, alkoxy, alkylthio, trifluoromethyl, trifluoromethoxy, trifluoromethylthio, nitro, cyano, amino, carboxy, phenoxy, benzyloxy, alkoxycarbonyl, alkylamino, dialkylamino, alkanoylamino, R² represents nitro, cyano, carbamoyl or -CONR⁵R⁶ or -NR⁶COR⁵ (wherein R⁵ is as hereinbefore defined for R¹ and R⁶ represents hydrogen or alkyl), R³ represents halogen, nitro, cyano, amino, carbamoyl, -CONR⁷R⁸ (wherein R⁷ is as hereinbefore defined for R¹ and R⁸ represents hydrogen or alkyl), and R⁴ represents hydrogen or alkyl, or salts thereof with the exclusion of compounds in which R² and R³ simultaneously represent cyano groups; plant-growth regulating compositions, novel compounds and their preparation are described.

摘要翻译： 本发明提供了使用下式化合物调节植物生长的方法：其中R 1表示任选被卤素，烷基，烷氧基，烷硫基，三氟甲基，三氟甲氧基，三氟甲硫基，硝基， 氰基，氨基，羧基，苯氧基，苄氧基，烷氧基羰基，烷基氨基，二烷基氨基，烷酰基氨基，R 2表示硝基，氰基，氨基甲酰基或-CONR 5 R 6或-NR 6 COR 5 R 5如上文定义，R 1和R 6代表氢或烷基），R 3表示卤素，硝基，氰基，氨基，氨基甲酰基，-CONR 7 R 8（其中 R 7如上文定义，R 1和R 8表示氢或烷基），R 4表示氢或烷基，或其盐，排除其中R 2和R 2的化合物 3同时表示氰基; 描述了植物生长调节组合物，新化合物及其制备方法。