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1.
公开(公告)号:EP0254105A2
公开(公告)日:1988-01-27
申请号:EP87109631.9
申请日:1987-07-03
申请人: MECT CORPORATION
发明人: Ogawa, Tomoya , Sugimott, Mamoru , Numata, Masaaki , Yoshimura, Shoji , Ito, Masayoshi , Shitori, Yoshiyasu
摘要: The present invention relates to sialic acid derivatives. According to the present invention, there is provided sialic acid derivatives having the general formula (I):
wherein, R 1 represents hydrogen, an acetyl group, a trityl group,
(R 5 represents hydrogen or an acetyl group and R 6 represents hydrogen, sodium or a methyl group). R 2 represents hydrogen or an acetyl group,
one of R 3 and R 4 represents chlorine, -OAc, -OH, -OCH 2 CH = CH 2 .
, or
(R 7 represents a hydrogen atom or an acetyl group, R 8 represents a hydrogen atom, an acetyl group or a benzyl group, R 9 represents a hydrogen atom, an acetyl group, a benzyl group or
or
wherein R 10 represents a hydrogen atom or a benzoyl group), while the other represents -COOR 11 wherein R" represents hydrogen, sodium, or a methyl group.摘要翻译: 本发明涉及唾液酸衍生物。 本发明提供具有通式(I)的唾液酸衍生物:
其中,R 1表示氢,乙酰基,三苯甲基,CHEM(R 5表示氢 或乙酰基,R 6表示氢,钠或甲基)。 R 2表示氢或乙酰基,R 3和R 4之一表示氯,-OAc,-OH,-OCH 2 CH = CH 2,CHEM或CHEM(R 7表示 氢原子或乙酰基,R 8表示氢原子,乙酰基或苄基,R 9表示氢原子,乙酰基,苄基或 ,其中R 1, <0>表示氢原子或苯甲酰基),而另一个表示-COOR 1,其中R 1表示氢,钠或甲基。 -
公开(公告)号:EP0254105A3
公开(公告)日:1988-04-20
申请号:EP87109631
申请日:1987-07-03
申请人: MECT CORPORATION
发明人: Ogawa, Tomoya , Sugimott, Mamoru , Numata, Masaaki , Yoshimura, Shoji , Ito, Masayoshi , Shitori, Yoshiyasu
摘要: The present invention relates to sialic acid derivatives. According to the present invention, there is provided sialic acid derivatives having the general formula (I):
wherein, R 1 represents hydrogen, an acetyl group, a trityl group,
(R 5 represents hydrogen or an acetyl group and R 6 represents hydrogen, sodium or a methyl group). R 2 represents hydrogen or an acetyl group, one of R 3 and R 4 represents chlorine, -OAc, -OH, -OCH 2 CH = CH 2 .
, or
(R 7 represents a hydrogen atom or an acetyl group, R 8 represents a hydrogen atom, an acetyl group or a benzyl group, R 9 represents a hydrogen atom, an acetyl group, a benzyl group or
or
wherein R 10 represents a hydrogen atom or a benzoyl group), while the other represents -COOR 11 wherein R" represents hydrogen, sodium, or a methyl group.
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