公开(公告)号：EP0172545A1

公开(公告)日：1986-02-26

申请号：EP85110331.7

申请日：1985-08-19

申请人： NIPPON KAYAKU CO., LTD.

发明人： Nakagawa, Taizo ,  Tanaka, Eiichi ,  Koike, Kengo ,  Yoshida, Hiromi ,  Yoshida, Hiroshi

IPC分类号： C07D213/81 ,  C07D213/82 ,  C07D405/12 ,  C07D409/12 ,  A01N43/40

CPC分类号： C07D213/81 ,  A01N43/40 ,  C07D213/82 ,  C07D405/12 ,  C07D409/12

摘要： Disclosed is the compound of the formula:

wherein X is oxygen, sulfur or


R, is 3-pyridyl or 4-pyridyl, R 2 is C 1 ~C 12 -alkyl; C 3 - or C 4 -alkenyl; C 5 - or C 6 -cycloalkyl which may be substituted by C,- or C 2 -alkyl; pyridyl; pyridylmethyl; phenethyl cyanoalkyl having 1 or 2 carbon atoms; methoxyethyl; 1-methylmethoxypropyl; phenyl; phenyl which is substituted by one or more of C 1 ~C 4 -alkyl, C 1 ~C 4 -alkoxy, nitro, halogen, trifluoromethyl, allyl and methoxycarbonyl; benzyl; benzyl which is substituted by one or more of methyl, nitro, methoxy and chloro; a-methylbenzyl; C 1 ~C 6 -alkyl which is substituted by halogen when X is oxygen or
C 2 - or C 3 -alkyl which is substituted by dimethylamino, furfuryl or thienylmethyl; R 3 is hydrogen, C 1 ~C 4 -alkyl, cyanomethyl, methoxycarbonylmethyl, or 1-propoxycarbonylmethyl.