-
1.发明授权STABLE CRYSTAL FORM OF 2-ETHYL-3, 7-DIMETHYL-6-(4-(TRIFLUOROMETHOXY) PHENOXY)QUINOLINE-4-YLMETHYL CARBONATE, METHOD OF MANUFACTURING SAME AND AGRICULTURAL CHEMICAL COMPOSITION CONTAINING CRYSTALS OF SAME 有权的2-乙基-3,7-二甲基-6-（4-（三氟甲氧基）苯氧基）稳定的结晶形式喹啉-4-基甲基碳酸酯，PROCESS AND THEREFOR农药组合物CRYSTAL THEREOF
公开(公告)号：EP2540709B1
公开(公告)日：2014-08-20
申请号：EP11747310.8
申请日：2011-02-22
发明人： TANIGAKIUCHI Kouki , SEKIGUCHI Mikio , HOTTA Hiroki , SHIMANO Shizuo , MORIKAWA Akinori , YAMAMOTO Kazumi , NAKANISHI Nozomu , MINOWA Nobuto , WATANABE Takashi
IPC分类号： C07D215/22 , A01N47/06 , A01P7/04
CPC分类号： C07D215/233 , A01N43/42 , A01N47/06 , C07D215/20 , A01N25/12
-
公开(公告)号：EP1240144A2
公开(公告)日：2002-09-18
申请号：EP00976295.6
申请日：2000-11-16
IPC分类号： C07D213/55 , C07D213/56 , C07D417/12 , A61K31/44 , A61P25/00
CPC分类号： C07D213/81 , C07C323/59 , C07D213/50 , C07D239/26 , C07D277/24 , C07D277/64 , C07D401/12 , C07D401/14 , C07D405/12 , C07D407/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D495/04
摘要： Neuroprotective agents are disclosed having structure: (I) and stereoisomers and pharmaceutically acceptable salts thereof, wherein R1 is alkyl, substituted alkyl, aryl, substituted aryl, arylalkyl, substituted arylalkyl, heterocycle, substituted heterocycle, heterocyclealkyl or substituted heterocyclealkyl; R2 is -OR2a or -NR2bR2c; R3 is hydrogen, keto, -C(=O)OR3a or -C(=O)NR3bR3c; R4 is hydrogen, alkyl, substituted alkyl, aryl, substituted aryl, -C(=O)R4a, -C(=O)OR4b, -C(=O)NR4cR4d, -OC(=O)NR4cR4d or -SO2R4c or wherein R3 and R4 taken together form a heterocyclic ring or substituted heterocyclic ring; and R5 is hydrogen, alkyl or substituted alkyl. Such compounds have utility in the treatment of conditions which benefit from administration of neuroprotective agents generally, including treatment of central and peripheral nervous condition as well as promoting nerve cell differentiation. Methods of treating such conditions are also disclosed, as are pharmaceutical compositions containing one or more of the compounds of this invention.
-
3.发明公开3-or 4-pyridinecarboxamide-derivates and their use as bactericides 失效3-或4- Pyridencarboxamidderivate以及它们作为杀菌剂的用途。
公开(公告)号：EP0172545A1
公开(公告)日：1986-02-26
申请号：EP85110331.7
申请日：1985-08-19
IPC分类号： C07D213/81 , C07D213/82 , C07D405/12 , C07D409/12 , A01N43/40
CPC分类号： C07D213/81 , A01N43/40 , C07D213/82 , C07D405/12 , C07D409/12
摘要： Disclosed is the compound of the formula:
wherein X is oxygen, sulfur or
R, is 3-pyridyl or 4-pyridyl, R 2 is C 1 ~C 12 -alkyl; C 3 - or C 4 -alkenyl; C 5 - or C 6 -cycloalkyl which may be substituted by C,- or C 2 -alkyl; pyridyl; pyridylmethyl; phenethyl cyanoalkyl having 1 or 2 carbon atoms; methoxyethyl; 1-methylmethoxypropyl; phenyl; phenyl which is substituted by one or more of C 1 ~C 4 -alkyl, C 1 ~C 4 -alkoxy, nitro, halogen, trifluoromethyl, allyl and methoxycarbonyl; benzyl; benzyl which is substituted by one or more of methyl, nitro, methoxy and chloro; a-methylbenzyl; C 1 ~C 6 -alkyl which is substituted by halogen when X is oxygen or
C 2 - or C 3 -alkyl which is substituted by dimethylamino, furfuryl or thienylmethyl; R 3 is hydrogen, C 1 ~C 4 -alkyl, cyanomethyl, methoxycarbonylmethyl, or 1-propoxycarbonylmethyl.-
公开(公告)号：EP3003709B1
公开(公告)日：2017-07-26
申请号：EP14726354.5
申请日：2014-05-23
发明人： TANAKA, Kouichi , FUJISAWA, Hideyoshi , IZUTANI, Kensuke , NISHIYAMA, Satoshi , TAKAMATSU, Atsushi , MATSUMOTO, Akira , FURUKAWA, Masayoshi
CPC分类号： G02B5/208 , B32B7/06 , B32B17/10036 , B32B17/10458 , B32B17/10633 , B32B17/10761 , B32B17/10788 , G02B5/0816 , G02B5/26 , G02B5/282 , G02B5/3016 , B32B17/10 , B32B2367/00
摘要： The present invention has the objective of providing an infrared reflective film by means of which it is possible to achieve an effective heat-shielding performance with a smaller number of layers than hitherto using a construction employing specified infrared reflective layers. Solution Means The infrared reflective film of the present invention has at least two infrared reflective layers and, of these infrared reflective layers, the center reflective wavelength of at least one infrared reflective layer is between 1200 and 1300 nm. Furthermore, the laminated glass of the present invention is formed by interposing this infrared reflective film between two sheets of intermediate film, and laminating these between two sheets of glass.
摘要翻译： 本发明的目的在于提供一种红外线反射膜，通过该红外线反射膜，与现有的使用特定的红外线反射层的结构相比，能够以更少的层数实现有效的隔热性能。 解决方案手段本发明的红外反射膜具有至少两个红外反射层，并且在这些红外反射层中，至少一个红外反射层的中心反射波长在1200和1300nm之间。 此外，本发明的夹层玻璃通过将该红外线反射膜夹在两片中间膜之间并将它们层压在两片玻璃之间而形成。
-
5.发明授权METHOD FOR PRODUCING 6-ARYLOXYQUINOLINE DERIVATIVE AND INTERMEDIATE THEREOF 有权用于生产6-ARYLOXYCHINOLIN衍生物和及其中间体
公开(公告)号：EP2305649B1
公开(公告)日：2013-04-24
申请号：EP09797889.4
申请日：2009-07-13
发明人： KATO Yasuhito , SHIMANO Shizuo , MORIKAWA Akinori , HOTTA Hiroki , YAMAMOTO Kazumi , NAKANISHI Nozomu , MINOWA Nobuto , KURIHARA Hiroshi
IPC分类号： C07D215/22 , C07C227/06 , C07C229/64 , C07B61/00
CPC分类号： C07D215/22 , C07C227/04 , C07C229/64 , C07D215/20
-
6.发明公开
公开(公告)号：EP2305649A1
公开(公告)日：2011-04-06
申请号：EP09797889.4
申请日：2009-07-13
发明人： KATO Yasuhito , SHIMANO Shizuo , MORIKAWA Akinori , HOTTA Hiroki , YAMAMOTO Kazumi , NAKANISHI Nozomu , MINOWA Nobuto , KURIHARA Hiroshi
IPC分类号： C07D215/22 , C07C227/06 , C07C229/64 , C07B61/00
CPC分类号： C07D215/22 , C07C227/04 , C07C229/64 , C07D215/20
摘要： Disclosed is a process for producing 6-aryloxyquinoline derivatives useful as insecticides or fungicides for agricultural and horticultural use. The process comprises a cyclization reaction step of reacting an anthranilic acid derivative represented by general formula (1) with a kenone in the presence of an acid to obtain a quinolone derivative and a condensation reaction step of reacting the quinolone derivative with a halogen compound or an acid anhydride to obtain a quinoline derivative.
摘要翻译： 披露了一种生产用作农业和园艺用杀虫剂或杀真菌剂的6-芳氧基喹啉衍生物的方法。 该方法包括使通式（1）所示的邻氨基苯甲酸衍生物与角鲨烯在酸存在下反应以获得喹诺酮衍生物的环化反应步骤和使喹诺酮衍生物与卤素化合物或卤素化合物反应的缩合反应步骤 酸酐反应得到喹啉衍生物。
-
7.发明公开MEDICINAL COMPOSITIONS FOR PREVENTING OR TREATING DIARRHEA 审中-公开医疗中心ZUSAMMENSETZUNGEN ZUR PREVENTION ODER BEHANDLUNG DERDIARRHÖ
公开(公告)号：EP1197214A1
公开(公告)日：2002-04-17
申请号：EP00942374.0
申请日：2000-06-28
发明人： TAKEUCHI, Tomio , MURAOKA, Yasuhiko , NISHIMURA, Yoshio , TERAYAMA, Yoshihiko Pharm. Techn. Labo , OKADA, Mineaki , AKIYAMA, Yuji , EKIMOTO, Hisao
IPC分类号： A61K31/7012 , A61P1/12
CPC分类号： C07H13/12 , A61K31/445 , A61K31/47 , A61K31/7012 , A61K45/06 , C07H7/02 , C07H13/04 , A61K2300/00
摘要： Provided is a pharmaceutical composition for the prevention or treatment of a diarrhea, which comprises as an active ingredient, siastatin B or a siastatin B derivative having a β-glucuronidase inhibitory activity. Siastatin B or the siastatin B derivative is useful as a drug for the prevention or treatment of a diarrhea, which is capable of ameliorating the diarrhea disorders as induced as a side effect when a cancer-bearing patient received the administration of an anticancer chemotherapeutic agent, particularly an anticancer camptothecin derivative acting as a topoisomerase I inhibitor. This composition is effective to prevent or treat such diarrhea as induced by the administration of an anticancer camptothecin derivative to the cancer-bearing patient.
摘要翻译： 提供了用于预防或治疗腹泻的药物组合物，其包含作为活性成分的具有β-葡糖醛酸糖苷酶抑制活性的西司特汀B或西司他丁B衍生物。 西塔他汀B或西沙星汀B衍生物可用作预防或治疗腹泻的药物，当患有癌症的患者接受抗癌化学治疗剂的施用时，其能够改善作为副作用诱导的腹泻病症， 特别是作为拓扑异构酶I抑制剂的抗癌喜树碱衍生物。 该组合物有效地预防或治疗由向抗癌患者施用抗癌喜树碱衍生物诱导的这种腹泻。
-
8.发明公开2,3-DISUBSTITUTED CYCLOPENTANONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND MEDICINAL USE THEREOF 失效2,3-二取代环戊酮衍生物，其医疗应用过程产生和
公开(公告)号：EP0976709A1
公开(公告)日：2000-02-02
申请号：EP97901810.8
申请日：1997-01-31
发明人： SAITO, Seiichi , MORINO, Tomio , MASUDA, Kuniko
IPC分类号： C07C49/517
CPC分类号： C07D213/80 , C07C49/517 , C07C62/26 , C07C323/22 , C07C323/41 , C07C323/59 , C07C2601/08 , C07D239/38 , C07D317/22 , C07D317/72
摘要： The present invention relates to a compound represented by the following general formula (1)
(wherein X represents O, S, SO, SO 2 , or NH, Y is a substituted or unsubstituted hydrocarbon residue containing 1 through 6 carbon atoms and having an overall molecular weight of not less than 15 and not more than 400, and the hydrocarbon residue, when the residue is ring, may contain one or two hetero-atoms in the ring, and Z is a carboxyl group , a group derived therefrom or an aliphatic hydrocarbon residue having from 1 to 4 carbon atoms which may be substituted or unsabstituted ) or a pharmacologically acceptable salt thereof (excluding (1R,2S)-2- [ (2R)-(2-acetylamino-2-carboxyethyl) thiomethyl ] -3-oxo-1-cyclopentanecarboxylic acid (cystacyclin)), a method for production thereof and a medicinal use thereof. The compound of the present invention is useful as a neuron differentiation accelerator.-
9.发明公开
公开(公告)号：EP3003709A1
公开(公告)日：2016-04-13
申请号：EP14726354.5
申请日：2014-05-23
发明人： TANAKA, Kouichi , FUJISAWA, Hideyoshi , IZUTANI, Kensuke , NISHIYAMA, Satoshi , TAKAMATSU, Atsushi , MATSUMOTO, Akira , FURUKAWA, Masayoshi
CPC分类号： G02B5/208 , B32B7/06 , B32B17/10036 , B32B17/10458 , B32B17/10633 , B32B17/10761 , B32B17/10788 , G02B5/0816 , G02B5/26 , G02B5/282 , G02B5/3016 , B32B17/10 , B32B2367/00
摘要： The present invention has the objective of providing an infrared reflective film by means of which it is possible to achieve an effective heat-shielding performance with a smaller number of layers than hitherto using a construction employing specified infrared reflective layers. Solution Means The infrared reflective film of the present invention has at least two infrared reflective layers and, of these infrared reflective layers, the center reflective wavelength of at least one infrared reflective layer is between 1200 and 1300 nm. Furthermore, the laminated glass of the present invention is formed by interposing this infrared reflective film between two sheets of intermediate film, and laminating these between two sheets of glass.
摘要翻译： 本发明的目的是提供一种红外线反射膜，通过该红外线反射膜，可以实现比迄今使用具有特定的红外线反射层的结构更少的层的有效的热屏蔽性能。 解决方案本发明的红外反射膜具有至少两个红外反射层，并且在这些红外反射层中，至少一个红外反射层的中心反射波长在1200和1300nm之间。 此外，本发明的夹层玻璃通过将这种红外反射膜插入两片中间膜之间并将它们层压在两片玻璃之间而形成。
-
10.发明授权
公开(公告)号：EP1780202B1
公开(公告)日：2013-02-27
申请号：EP05768511.7
申请日：2005-08-03
发明人： YAMAMOTO, Kazumi , HORIKOSHI, Ryo , OYAMA, Kazuhiko , KURIHARA, Hiroshi , SHIMANO, Shizuo , MIYAKE, Takaaki , HOTTA, Hiroki , IWABUCHI, Jun
IPC分类号： C07D215/22 , A01N25/04 , A01N25/12 , A01N25/14 , A01N43/42 , C07D215/36
CPC分类号： C07D215/233 , A01N43/42 , C07D215/36
-
-
-
-
-
-
-
-
-
搜索结果
27 条记录 (耗时 0.02 秒)
