公开(公告)号：EP1031567B1

公开(公告)日：2003-04-02

申请号：EP98950461.8

申请日：1998-10-30

申请人： Nihon Nohyaku Co., Ltd.

发明人： TSUBATA, Kenji ,  SANPEI, Osamu ,  TAKAGI, Kazuhiro ,  UMETANI, Kunihisa ,  UCHIKUROHANE, Tohru ,  TAJIMA, Sohkichi

IPC分类号： C07D285/06 ,  A01N43/82

CPC分类号： C07D285/06 ,  A01N43/82

摘要： N-(3-Chloro-4-methylphenyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide; a plant disease controlling agent characterized by containing the compound as the active ingredient; and a method of using the same. The agent is excellent in the activity of controlling plant diseases such as blast.

公开(公告)号：EP3043791A1

公开(公告)日：2016-07-20

申请号：EP14781682.1

申请日：2014-09-12

申请人： Nihon Nohyaku Co., Ltd. ,  Pitney Pharmaceuticals Pty Limited

发明人： ANDOH, Nobuharu ,  SANPEI, Osamu ,  TOGA, Tetsuo ,  MORRIS, David Lawson ,  ASTON, Roger ,  TANAKA, Koji ,  HINO, Tomokazu

IPC分类号： A61K31/277 ,  A61K31/415 ,  A61P35/00

CPC分类号： A61K31/277 ,  A61K31/341 ,  A61K31/381 ,  A61K31/415 ,  A61K31/4196 ,  A61K31/42 ,  A61K31/421 ,  A61K31/4245 ,  A61K31/426 ,  A61K31/433 ,  A61K31/437 ,  A61K31/44 ,  A61K31/4965 ,  A61K31/505 ,  A61K31/5377 ,  A61K31/5383

摘要： wherein R1 is a hydrogen atom, an alkyl group and the like, R2, R3, and R4 are the same or different and each is a hydrogen atom, an alkyl group and the like, R5 and R6 are the same or different and each is a hydrogen atom, a halogen atom and the like, m is 0 or 1, R is a halogen atom, a cyano group, a nitro group, a phenyl group optionally substituted by an alkyl group and the like, an alkyl group and the like, Ar1 is a phenyl group, a naphthyl group, a pyridyl group, a pyrazolyl group, or the like, each of which is optionally substituted by a halogen atom, a cyano group, a nitro group, alkyl group and the like, and W is —O—, —S—, —SO2—, or —N(R7)—wherein R7 is a hydrogen atom, a (C1-C6) alkyl group and the like, or a pharmacologically acceptable salt thereof.

公开(公告)号：EP1216988A1

公开(公告)日：2002-06-26

申请号：EP00962896.7

申请日：2000-09-27

申请人： Nihon Nohyaku Co., Ltd.

发明人： SANPEI, Osamu ,  TSUBATA, Kenji

IPC分类号： C07C323/25 ,  C07D213/70 ,  C07D295/08 ,  C07D333/34 ,  C07D213/89 ,  C07C319/14

CPC分类号： C07D213/70 ,  C07C323/25 ,  C07C2601/08 ,  C07D213/89 ,  C07D249/12 ,  C07D295/088 ,  C07D333/34

摘要： The present invention relates to a thioalkylamine derivative represented by general formula (I); and a process for production thereof:
wherein each of R 1 and R 2 is H, (C 1 -C 4 )alkyl, (C 3 -C 8 )cycloalkyl, (C 3 -C 8 )cycloalkyl (C 1 -C 4 ) alkyl, (substituted) phenyl, (substituted) phenyl(C 1 -C 4 ) alkyl, or the like; each of R 3 and R 4 is H or a (C 1 -C 4 )alkyl group; each of R 5 and R 6 is H, (C 1 -C 4 )alkyl, a (substituted) phenyl group or a (substituted) phenyl(C 1 -C 4 )alkyl group; alternatively each of R 1 and R 2 , R 1 and R 3 or R 5 , R 3 and R 4 , R 3 and R 5 , or R 5 and R 6 may together form lower alkylene; and R is (C 1 -C 12 )alkyl, (C 3 -C 8 )cycloalkyl, (C 3 -C 8 )cycloalkyl (C 1 -C 4 ) alkyl, (substituted) phenyl, (substituted) phenyl (C 1 -C 4 )alkyl, a naphthyl group, a (substituted) aromatic heterocyclic, or the like.

摘要翻译： 本发明涉及由通式（I）表示的硫烷基胺衍生物。 及其制备方法：其中R 1和R 2各自为H，（C 1 -C 4）烷基，（C 3 -C 8）环烷基，（C 3 -C 8）环烷基（C 1 -C 4）烷基，（取代的） ，（取代的）苯基（C 1 -C 4）烷基等; R 3和R 4各自为H或（C 1 -C 4）烷基; R5和R6各自为H，（C1-C4）烷基，（取代）苯基或（取代）苯基（C1-C4）烷基; 或者R1和R2中的每一个，R 1和R 3或R 5，R 3和R 4，R 3和R 5或R 5和R 6可以一起形成低级亚烷基; （C 1 -C 4）烷基，（C 3 -C 8）环烷基，（C 3 -C 8）环烷基（C 1 -C 4）烷基，（取代的）苯基，（取代的） （取代的）芳族杂环基等。

公开(公告)号：EP1031567A1

公开(公告)日：2000-08-30

申请号：EP98950461.8

申请日：1998-10-30

申请人： Nihon Nohyaku Co., Ltd.

发明人： TSUBATA, Kenji ,  SANPEI, Osamu ,  TAKAGI, Kazuhiro ,  UMETANI, Kunihisa ,  UCHIKUROHANE, Tohru ,  TAJIMA, Sohkichi

IPC分类号： C07D285/06 ,  A01N43/82

CPC分类号： C07D285/06 ,  A01N43/82

摘要： The present invention relates to N-(3-chloro-4-methylphenyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide, a plant disease controller characterized by containing said compound as an active ingredient, and a usage of said plant disease controller. The plant disease controller of the present invention has an excellent controlling activity against plant diseases such as blast.

摘要翻译： 本发明涉及N-（3-氯-4-甲基 - 苯基）-4-甲基-1,2,3-噻二唑-5-甲酰胺，通过在含有所述化合物作为活性成分为特征的植物病害防治剂，以及使用 所述植物病害防治剂的。 本发明的植物病害防治剂在对植物病害具有出色的控制活性：如爆炸。